Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Methionine aminopeptidase 1 (Homo sapiens (Human)) | BDBM50558959 (CHEMBL4740594) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111860 BindingDB Entry DOI: 10.7270/Q24171R4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase 1 (Homo sapiens (Human)) | BDBM50558957 (CHEMBL4755128) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111860 BindingDB Entry DOI: 10.7270/Q24171R4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase 1 (Homo sapiens (Human)) | BDBM50558956 (CHEMBL4743733) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111860 BindingDB Entry DOI: 10.7270/Q24171R4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase 1 (Homo sapiens (Human)) | BDBM50558967 (CHEMBL4759563) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111860 BindingDB Entry DOI: 10.7270/Q24171R4 | |||||||||||
More data for this Ligand-Target Pair |