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Compile Data Set for Download or QSAR

Found 4 hits of kd for UniProtKB: P53582   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Methionine aminopeptidase 1


(Homo sapiens (Human))
BDBM50558959
PNG
(CHEMBL4740594)
Show SMILES Oc1cccc2ccc(nc12)C1SCC(=O)N1c1cccc(F)c1
PDB
MMDB

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UniProtKB/SwissProt

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DrugBank
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GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/a 1.5n/an/an/an/an/a


TBA

Assay Description
Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis


Citation and Details

Article DOI: 10.1016/j.ejmech.2019.111860
BindingDB Entry DOI: 10.7270/Q24171R4
More data for this
Ligand-Target Pair
Methionine aminopeptidase 1


(Homo sapiens (Human))
BDBM50558957
PNG
(CHEMBL4755128)
Show SMILES Oc1cccc2ccc(nc12)C1SCC(=O)N1c1cccc(c1)C#N
PDB
MMDB

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UniProtKB/SwissProt

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DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/a 3.5n/an/an/an/an/a


TBA

Assay Description
Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis


Citation and Details

Article DOI: 10.1016/j.ejmech.2019.111860
BindingDB Entry DOI: 10.7270/Q24171R4
More data for this
Ligand-Target Pair
Methionine aminopeptidase 1


(Homo sapiens (Human))
BDBM50558956
PNG
(CHEMBL4743733)
Show SMILES Oc1cccc2ccc(nc12)C1SCC(=O)N1c1ccc(Cl)cc1
PDB
MMDB

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UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/a 3.60n/an/an/an/an/a


TBA

Assay Description
Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis


Citation and Details

Article DOI: 10.1016/j.ejmech.2019.111860
BindingDB Entry DOI: 10.7270/Q24171R4
More data for this
Ligand-Target Pair
Methionine aminopeptidase 1


(Homo sapiens (Human))
BDBM50558967
PNG
(CHEMBL4759563)
Show SMILES Cc1ccc(cc1)N1C(SCC1=O)c1ccc2cccc(O)c2n1
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/a 8.5n/an/an/an/an/a


TBA

Assay Description
Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysis


Citation and Details

Article DOI: 10.1016/j.ejmech.2019.111860
BindingDB Entry DOI: 10.7270/Q24171R4
More data for this
Ligand-Target Pair