Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucocorticoid receptor (MOUSE) | BDBM50016932 (CHEMBL3273976) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrs | J Med Chem 20: 1134-9 (1978) BindingDB Entry DOI: 10.7270/Q2RX9DM6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (MOUSE) | BDBM13775 ((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid PDB UniChem Similars | PDB PubMed | n/a | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrs | J Med Chem 20: 1134-9 (1978) BindingDB Entry DOI: 10.7270/Q2RX9DM6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glucocorticoid receptor (MOUSE) | BDBM50016931 (CHEBI:31677 | HYDROCORTISONE HEMISUCCINATE | Hydro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrs | J Med Chem 20: 1134-9 (1978) BindingDB Entry DOI: 10.7270/Q2RX9DM6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (MOUSE) | BDBM50016933 (CHEMBL3273977) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 430 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrs | J Med Chem 20: 1134-9 (1978) BindingDB Entry DOI: 10.7270/Q2RX9DM6 | |||||||||||
More data for this Ligand-Target Pair |