Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ecdysone receptor (Bombyx mori) | BDBM50488465 (CHEMBL2286413) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.24E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488464 (CHEMBL2286419) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.91E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488463 (CHEMBL2285681) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.35E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488437 (CHEMBL2286416) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.48E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488438 (CHEMBL2286414) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488477 (CHEMBL2286417) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.69E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488448 (CHEMBL2286411) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.82E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488462 (CHEMBL2286415) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.79E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ecdysone receptor (Bombyx mori) | BDBM50488447 (CHEMBL2286412) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.76E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge... | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
More data for this Ligand-Target Pair |