Compile Data Set for Download or QSAR

Found 10 hits of ic50 for UniProtKB: P0C7A3   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548065 (CHEMBL4785875) Show SMILES Cc1nc(ccc1COc1cc(Cl)c2cc(CC(O)=O)sc2c1Cl)C(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548066 (CHEMBL4791105) Show SMILES OC(=O)c1ccc2oc(SCc3ccc(Cl)cc3Cl)nc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548069 (CHEMBL4741670) Show SMILES CCCC[C@H]1C[C@@H](C1)C(=O)NC[C@H]1CCCN1C(=O)[C@@H](NC(=S)CNC)C(C)(C)C |r,wU:12.12,6.8,wD:19.27,4.3,(17.81,-5.97,;17.5,-7.47,;18.64,-8.5,;20.11,-8.02,;21.25,-9.05,;21.33,-10.59,;22.86,-10.5,;22.79,-8.97,;24.01,-11.53,;25.48,-11.05,;23.69,-13.04,;24.84,-14.07,;24.52,-15.57,;25.55,-16.72,;24.78,-18.05,;23.28,-17.73,;23.11,-16.21,;21.77,-15.44,;21.77,-13.9,;20.44,-16.21,;19.11,-15.44,;17.77,-16.21,;17.77,-17.75,;16.44,-15.44,;15.1,-16.21,;13.77,-15.44,;20.44,-17.75,;19.11,-18.52,;21.77,-18.52,;20.42,-19.28,)| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548072 (CHEMBL4778987) Show SMILES CCCCCCCC(=O)NC[C@H](NC(=O)[C@H](CO)NC(=O)CN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CN)CC(C)C |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	KEGG PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548074 (CHEMBL4750990) Show SMILES CCCCCCCC(=O)OC[C@H](OC(=O)[C@H](CO)NC(=O)CN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCNC(N)=N)C(O)=O |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	KEGG PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548068 (CHEMBL4753228) Show SMILES CCCCCCN(C(CNCc1ccccc1)c1ccc2cc(O)ccc2c1)C(C)=O Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548067 (CHEMBL4762372) Show SMILES CCCCCCCCN(C(CNCc1ccccc1)c1ccc2cc(O)ccc2c1)C(C)=O Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548073 (CHEMBL4756686) Show SMILES CCCCCCCC(=O)OC[C@H](NC(=O)[C@H](CO)NC(=O)CN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CN)CC(C)C |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548070 (CHEMBL4784392) Show SMILES CCCCCCC[C@](C)(O)\C=C\[C@H](NC(=O)OCc1ccccc1)C(=O)OC |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548071 (CHEMBL4788110) Show SMILES CCCCCCC[C@H](O)\C=C\[C@H](NC(=O)OCc1ccccc1)C(=O)OC |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	9.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair