Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein disulfide-isomerase A4 (Homo sapiens) | BDBM50550835 (CHEMBL4751979) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.31E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assay | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111906 BindingDB Entry DOI: 10.7270/Q2125X88 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein disulfide-isomerase A4 (Homo sapiens) | BDBM50550836 (CHEMBL4751241) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.16E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assay | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111906 BindingDB Entry DOI: 10.7270/Q2125X88 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein disulfide-isomerase A4 (Homo sapiens) | BDBM50550837 (CHEMBL4762045) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assay | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111906 BindingDB Entry DOI: 10.7270/Q2125X88 | |||||||||||
More data for this Ligand-Target Pair |