Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gamma-aminobutyric acid receptor subunit beta-1 (Homo sapiens (Human)) | BDBM50581248 (CHEMBL5090753) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human GABAB1b receptor expressed in RBL cells by microplate analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00802 BindingDB Entry DOI: 10.7270/Q2542SG3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462446 (CHEMBL4238634) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.94E+4 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462450 (CHEMBL4238712) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.27E+4 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50427613 (CHEMBL2322935) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462443 (CHEMBL4238315) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.74E+4 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462444 (CHEMBL4244129) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.10E+4 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462449 (CHEMBL4247210) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462445 (CHEMBL4246158) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462451 (CHEMBL4249205) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462447 (CHEMBL4248377) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462453 (CHEMBL4244933) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462454 (CHEMBL4250786) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462442 (CHEMBL4245403) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462448 (CHEMBL4241188) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit beta-1/beta-2 (Homo sapiens (Human)) | BDBM50462452 (CHEMBL4244940) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte... | Bioorg Med Chem Lett 28: 2697-2700 (2018) Article DOI: 10.1016/j.bmcl.2018.04.003 BindingDB Entry DOI: 10.7270/Q20P12N7 | |||||||||||
More data for this Ligand-Target Pair |