Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463126 (CHEMBL4238599) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to His-tagged Myc (unknown origin) expressed in Escherichia coli BL21 by Bio-FET analysis | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463128 (CHEMBL4249055) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to His-tagged Myc (unknown origin) expressed in Escherichia coli BL21 by Bio-FET analysis | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50423921 (CHEMBL2312756) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a |
University of Maryland Curated by ChEMBL | Assay Description Binding affinity to human c-Myc bHLH-ZIP domain (353 to 437 amino acid residues) expressed in Escherichia coli BL21 (DE3) by fluorescence polarizatio... | Bioorg Med Chem Lett 23: 370-4 (2012) Article DOI: 10.1016/j.bmcl.2012.10.013 BindingDB Entry DOI: 10.7270/Q2WM1FPM | |||||||||||
More data for this Ligand-Target Pair |