Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential cation channel subfamily V member 1 (Mus musculus) | BDBM50539315 (CHEMBL4648896) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Seoul National University Curated by ChEMBL | Assay Description Antagonist activity at capsaicin-induced mouse TRPV1 expressed in CHOK1 cells by FLIPR assay | Bioorg Med Chem Lett 30: (2020) Article DOI: 10.1016/j.bmcl.2019.126838 BindingDB Entry DOI: 10.7270/Q2VD730D | |||||||||||
More data for this Ligand-Target Pair |