Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Solute carrier family 15 member 1 (Rattus norvegicus) | BDBM50344967 (2-[(4-Isopropyl-cyclohexanecarbonyl)-amino]-3-phen...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University Hospital Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 20 uM) in PEPT1-expressing LLC-PK1 cells | Eur J Pharmacol 392: 11-7 (2000) Article DOI: 10.1016/s0014-2999(00)00119-9 BindingDB Entry DOI: 10.7270/Q2HH6NXP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 15 member 1 (Rattus norvegicus) | BDBM5025 (Oseltamivir | US10919856, POSITIVE CONTROL | ethyl...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.83E+7 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Michigan Curated by ChEMBL | Assay Description Inhibition of rat recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation c... | Drug Metab Dispos 40: 1328-35 (2012) Article DOI: 10.1124/dmd.111.044263 BindingDB Entry DOI: 10.7270/Q2DZ0B1K | |||||||||||
More data for this Ligand-Target Pair |