Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteasome subunit alpha type-1 (Homo sapiens (Human)) | BDBM50577134 (CHEMBL4877708) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113556 BindingDB Entry DOI: 10.7270/Q2BR8WZN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-1 (Homo sapiens (Human)) | BDBM50577116 (CHEMBL4872258) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.36E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113556 BindingDB Entry DOI: 10.7270/Q2BR8WZN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-1 (Homo sapiens (Human)) | BDBM50577133 (CHEMBL4870115) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113556 BindingDB Entry DOI: 10.7270/Q2BR8WZN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-1 (Homo sapiens (Human)) | BDBM50577131 (CHEMBL4855915) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113556 BindingDB Entry DOI: 10.7270/Q2BR8WZN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-1 (Homo sapiens (Human)) | BDBM50007203 (CHEMBL3237875) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113556 BindingDB Entry DOI: 10.7270/Q2BR8WZN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-1 (Homo sapiens (Human)) | BDBM50577130 (CHEMBL4846410) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113556 BindingDB Entry DOI: 10.7270/Q2BR8WZN | |||||||||||
More data for this Ligand-Target Pair |