Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-1 adrenergic receptor (Mus musculus) | BDBM50225512 (CHEMBL157187) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) binding | J Med Chem 28: 634-42 (1985) BindingDB Entry DOI: 10.7270/Q2PN97VW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Mus musculus) | BDBM50225513 (CHEMBL423055) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) binding in SF-49 lymphoma cell | J Med Chem 28: 634-42 (1985) BindingDB Entry DOI: 10.7270/Q2PN97VW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Mus musculus) | BDBM50225514 (CHEMBL160277) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) binding | J Med Chem 28: 634-42 (1985) BindingDB Entry DOI: 10.7270/Q2PN97VW | |||||||||||
More data for this Ligand-Target Pair |