Found 135 hits of ic50 for UniProtKB: P09217 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kcal/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50468260
(CHEMBL4282837)Show SMILES [H][C@]12C[C@@H](NC)[C@@H](OC)[C@](C)(O1)n1c3ccc(O)cc3c3c4CNC(=O)c4c4c5cc(O)ccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O5/c1-28-26(36-3)17(29-2)10-20(37-28)31-18-6-4-12(33)8-14(18)22-23-16(11-30-27(23)35)21-15-9-13(34)5-7-19(15)32(28)25(21)24(22)31/h4-9,17,20,26,29,33-34H,10-11H2,1-3H3,(H,30,35)/t17-,20-,26-,28+/m1/s1 | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
PAK Research Center
Curated by ChEMBL
| Assay Description
Inhibition of rat brain PKC using RGFR derived peptide substrate |
Eur J Med Chem 142: 229-243 (2017)
Article DOI: 10.1016/j.ejmech.2017.07.043
BindingDB Entry DOI: 10.7270/Q21J9DG3 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469649
(CHEMBL283259)Show SMILES O=C1NC(=O)c2c1c1c3ccccc3n3CS(=O)(=O)Cn4c5ccccc5c2c4c13 Show InChI InChI=1S/C22H13N3O4S/c26-21-17-15-11-5-1-3-7-13(11)24-9-30(28,29)10-25-14-8-4-2-6-12(14)16(20(25)19(15)24)18(17)22(27)23-21/h1-8H,9-10H2,(H,23,26,27) | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469642
(CHEMBL282805)Show SMILES CC1n2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(C(C)S1(=O)=O)c4c23 Show InChI InChI=1S/C24H17N3O4S/c1-11-26-15-9-5-3-7-13(15)17-19-20(24(29)25-23(19)28)18-14-8-4-6-10-16(14)27(22(18)21(17)26)12(2)32(11,30)31/h3-12H,1-2H3,(H,25,28,29) | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469642
(CHEMBL282805)Show SMILES CC1n2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(C(C)S1(=O)=O)c4c23 Show InChI InChI=1S/C24H17N3O4S/c1-11-26-15-9-5-3-7-13(15)17-19-20(24(29)25-23(19)28)18-14-8-4-6-10-16(14)27(22(18)21(17)26)12(2)32(11,30)31/h3-12H,1-2H3,(H,25,28,29) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1 | PDB
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MCE
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| Article
PubMed
| n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cephalon, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C |
J Med Chem 40: 2994-6 (1997)
Article DOI: 10.1021/jm9702037
BindingDB Entry DOI: 10.7270/Q2377CF0 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469644
(CHEMBL281448)Show SMILES O=C1NCc2c1c1c3ccccc3n3CS(=O)(=O)Cn4c5ccccc5c2c4c13 Show InChI InChI=1S/C22H15N3O3S/c26-22-19-14(9-23-22)17-12-5-1-3-7-15(12)24-10-29(27,28)11-25-16-8-4-2-6-13(16)18(19)21(25)20(17)24/h1-8H,9-11H2,(H,23,26) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1 | PDB
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TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469655
(CHEMBL26872)Show InChI InChI=1S/C22H15N3OS/c26-22-19-14(9-23-22)17-12-5-1-3-7-15(12)24-10-27-11-25-16-8-4-2-6-13(16)18(19)21(25)20(17)24/h1-8H,9-11H2,(H,23,26) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
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| Article
| n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469652
(CHEMBL285613)Show SMILES OCC(CO)N1Cn2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(C1)c4c23 Show InChI InChI=1S/C25H20N4O4/c30-9-13(10-31)27-11-28-16-7-3-1-5-14(16)18-20-21(25(33)26-24(20)32)19-15-6-2-4-8-17(15)29(12-27)23(19)22(18)28/h1-8,13,30-31H,9-12H2,(H,26,32,33) | PDB
UniProtKB/SwissProt
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| PC cid
PC sid
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| Article
| n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1 | PDB
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| n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C |
Bioorg Med Chem Lett 9: 2279-82 (1999)
BindingDB Entry DOI: 10.7270/Q2MW2K90 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469643
(CHEMBL284632)Show SMILES O=C1NC(=O)c2c1c1c3ccccc3n3COCn4c5ccccc5c2c4c13 Show InChI InChI=1S/C22H13N3O3/c26-21-17-15-11-5-1-3-7-13(11)24-9-28-10-25-14-8-4-2-6-12(14)16(20(25)19(15)24)18(17)22(27)23-21/h1-8H,9-10H2,(H,23,26,27) | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469641
(CHEMBL283903)Show SMILES O=C1NC(=O)c2c1c1c3ccccc3n3CSCn4c5ccccc5c2c4c13 Show InChI InChI=1S/C22H13N3O2S/c26-21-17-15-11-5-1-3-7-13(11)24-9-28-10-25-14-8-4-2-6-12(14)16(20(25)19(15)24)18(17)22(27)23-21/h1-8H,9-10H2,(H,23,26,27) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469640
(CHEMBL26817)Show SMILES OCCN1Cn2c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n(C1)c4c23 Show InChI InChI=1S/C24H20N4O2/c29-10-9-26-12-27-17-7-3-1-5-14(17)19-16-11-25-24(30)21(16)20-15-6-2-4-8-18(15)28(13-26)23(20)22(19)27/h1-8,29H,9-13H2,(H,25,30) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469645
(CHEMBL26074)Show SMILES OCCN1Cn2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(C1)c4c23 Show InChI InChI=1S/C24H18N4O3/c29-10-9-26-11-27-15-7-3-1-5-13(15)17-19-20(24(31)25-23(19)30)18-14-6-2-4-8-16(14)28(12-26)22(18)21(17)27/h1-8,29H,9-12H2,(H,25,30,31) | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50478518
(CHEMBL514017)Show SMILES [H][C@]12[C@]3([H])C=C(CO)C[C@]4(O)C(=O)C(C)=C[C@@]4([H])[C@@]3(O)[C@@H](C)C[C@@]1(OC(=O)C\C=C\C=C\CCCC)C2(C)C |r,c:14,t:4| Show InChI InChI=1S/C30H42O6/c1-6-7-8-9-10-11-12-13-24(32)36-29-16-20(3)30(35)22(25(29)27(29,4)5)15-21(18-31)17-28(34)23(30)14-19(2)26(28)33/h9-12,14-15,20,22-23,25,31,34-35H,6-8,13,16-18H2,1-5H3/b10-9+,12-11+/t20-,22-,23+,25+,28+,29-,30+/m0/s1 | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
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| Article
PubMed
| n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute
Curated by ChEMBL
| Assay Description
Displacement of [3H]PDBu from rat brain membrane PKC |
J Nat Prod 58: 769-72 (1995)
Article DOI: 10.1021/np50119a020
BindingDB Entry DOI: 10.7270/Q2NZ8BF5 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469646
(CHEMBL27387)Show SMILES [O-][S+]1Cn2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(C1)c4c23 Show InChI InChI=1S/C22H13N3O3S/c26-21-17-15-11-5-1-3-7-13(11)24-9-29(28)10-25-14-8-4-2-6-12(14)16(20(25)19(15)24)18(17)22(27)23-21/h1-8H,9-10H2,(H,23,26,27) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
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| Article
| n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469650
(CHEMBL283399)Show SMILES O=C1NC(=O)c2c1c1c3ccccc3n3C4COCC(n5c6ccccc6c2c5c13)S4(=O)=O Show InChI InChI=1S/C24H15N3O5S/c28-23-19-17-11-5-1-3-7-13(11)26-15-9-32-10-16(33(15,30)31)27-14-8-4-2-6-12(14)18(22(27)21(17)26)20(19)24(29)25-23/h1-8,15-16H,9-10H2,(H,25,28,29) | PDB
UniProtKB/SwissProt
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| PC cid
PC sid
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| Article
| n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469639
(CHEMBL282298)Show SMILES CCOC(=O)C1n2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(CS1(=O)=O)c4c23 Show InChI InChI=1S/C25H17N3O6S/c1-2-34-25(31)24-28-15-10-6-4-8-13(15)17-19-18(22(29)26-23(19)30)16-12-7-3-5-9-14(12)27(11-35(24,32)33)20(16)21(17)28/h3-10,24H,2,11H2,1H3,(H,26,29,30) | PDB
UniProtKB/SwissProt
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| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469653
(CHEMBL282612)Show SMILES NC1=NC(=O)c2c1c1c3ccccc3n3CSCn4c5ccccc5c2c4c13 |t:1| Show InChI InChI=1S/C22H14N4OS/c23-21-17-15-11-5-1-3-7-13(11)25-9-28-10-26-14-8-4-2-6-12(14)16(20(26)19(15)25)18(17)22(27)24-21/h1-8H,9-10H2,(H2,23,24,27) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469647
(CHEMBL283930)Show SMILES NC1=NC(=O)c2c1c1c3ccccc3n3COCn4c5ccccc5c2c4c13 |t:1| Show InChI InChI=1S/C22H14N4O2/c23-21-17-15-11-5-1-3-7-13(11)25-9-28-10-26-14-8-4-2-6-12(14)16(20(26)19(15)25)18(17)22(27)24-21/h1-8H,9-10H2,(H2,23,24,27) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
| Article
| n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50478561
(CHEBI:69599 | Methylpendolmycin)Show SMILES [H][C@@]1([C@@H](C)CC)N(C)c2ccc(c3[nH]cc(C[C@@H](CO)NC1=O)c23)C(C)(C)C=C |r| Show InChI InChI=1S/C23H33N3O2/c1-7-14(3)21-22(28)25-16(13-27)11-15-12-24-20-17(23(4,5)8-2)9-10-18(19(15)20)26(21)6/h8-10,12,14,16,21,24,27H,2,7,11,13H2,1,3-6H3,(H,25,28)/t14-,16-,21-/m0/s1 | PDB
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| Article
PubMed
| n/a | n/a | 35.2 | n/a | n/a | n/a | n/a | n/a | n/a |
Sterling Research Group
Curated by ChEMBL
| Assay Description
Displacement of radiolabeled PDBU from PKC in rat forebrain |
J Nat Prod 54: 1440-3
Article DOI: 10.1021/np50077a040
BindingDB Entry DOI: 10.7270/Q2377CGF |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM6760
((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)Show SMILES COC(=O)[C@@]1(O)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C27H21N3O5/c1-26-27(33,25(32)34-2)11-18(35-26)29-16-9-5-3-7-13(16)20-21-15(12-28-24(21)31)19-14-8-4-6-10-17(14)30(26)23(19)22(20)29/h3-10,18,33H,11-12H2,1-2H3,(H,28,31)/t18?,26-,27-/m0/s1 | PDB
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| n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50241867
(((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...)Show SMILES C[C@@H]1O[C@@H](O[C@@H]2[C@@H](O)[C@H](OCCc3ccc(O)c(O)c3)O[C@H](CO)[C@H]2OC(=O)\C=C\c2ccc(O)c(O)c2)[C@H](O)[C@H](O)[C@H]1O |r| Show InChI InChI=1S/C29H36O15/c1-13-22(36)23(37)24(38)29(41-13)44-27-25(39)28(40-9-8-15-3-6-17(32)19(34)11-15)42-20(12-30)26(27)43-21(35)7-4-14-2-5-16(31)18(33)10-14/h2-7,10-11,13,20,22-34,36-39H,8-9,12H2,1H3/b7-4+/t13-,20+,22-,23+,24+,25+,26+,27+,28+,29-/m0/s1 | PDB
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| n/a | n/a | 68 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi Recherche
Curated by ChEMBL
| Assay Description
Displacement of [3H]PDBu from rat brain PKC by scintillation counting |
J Nat Prod 54: 1595-600
Article DOI: 10.1021/np50078a016
BindingDB Entry DOI: 10.7270/Q23T9KWX |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469654
(CHEMBL28202)Show SMILES CN1Cn2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(C1)c4c23 Show InChI InChI=1S/C23H16N4O2/c1-25-10-26-14-8-4-2-6-12(14)16-18-19(23(29)24-22(18)28)17-13-7-3-5-9-15(13)27(11-25)21(17)20(16)26/h2-9H,10-11H2,1H3,(H,24,28,29) | PDB
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| n/a | n/a | 86 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469651
(CHEMBL26996)Show SMILES ON1Cn2c3ccccc3c3c4C(=O)NC(=O)c4c4c5ccccc5n(C1)c4c23 Show InChI InChI=1S/C22H14N4O3/c27-21-17-15-11-5-1-3-7-13(11)25-9-24(29)10-26-14-8-4-2-6-12(14)16(20(26)19(15)25)18(17)22(28)23-21/h1-8,29H,9-10H2,(H,23,27,28) | PDB
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| n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50469648
(CHEMBL26936)Show SMILES O=C1NC(=O)c2c1c1c3ccccc3n3CNCn4c5ccccc5c2c4c13 Show InChI InChI=1S/C22H14N4O2/c27-21-17-15-11-5-1-3-7-13(11)25-9-23-10-26-14-8-4-2-6-12(14)16(20(26)19(15)25)18(17)22(28)24-21/h1-8,23H,9-10H2,(H,24,27,28) | PDB
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| n/a | n/a | 145 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
In vitro inhibition of protein kinase C from rat brain. |
Citation and Details
Article DOI: 10.1016/S0960-894X(01)80356-5
BindingDB Entry DOI: 10.7270/Q25M68DB |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM6760
((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)Show SMILES COC(=O)[C@@]1(O)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C27H21N3O5/c1-26-27(33,25(32)34-2)11-18(35-26)29-16-9-5-3-7-13(16)20-21-15(12-28-24(21)31)19-14-8-4-6-10-17(14)30(26)23(19)22(20)29/h3-10,18,33H,11-12H2,1-2H3,(H,28,31)/t18?,26-,27-/m0/s1 | PDB
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| n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Cephalon, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C |
J Med Chem 40: 2994-6 (1997)
Article DOI: 10.1021/jm9702037
BindingDB Entry DOI: 10.7270/Q2377CF0 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50217039
(CHEMBL420938)Show InChI InChI=1S/C14H10O2S3/c15-6-9-5-14(17-8-9)13-4-3-12(19-13)11-2-1-10(7-16)18-11/h1-5,7-8,15H,6H2 | PDB
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| n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C |
Bioorg Med Chem Lett 9: 2279-82 (1999)
BindingDB Entry DOI: 10.7270/Q2MW2K90 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1 | PDB
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| n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Tokyo University of Agriculture
Curated by ChEMBL
| Assay Description
Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of mouse anti-DNP IgE-stimulated beta-hexosaminidase release preincubated for 15 mins fo... |
Bioorg Med Chem Lett 30: (2020)
Article DOI: 10.1016/j.bmcl.2019.126886
BindingDB Entry DOI: 10.7270/Q26Q21RR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1 | PDB
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| n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Tokyo University of Agriculture
Curated by ChEMBL
| Assay Description
Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of anti-DNP IgE-stimulated TNFalpha release preincubated for 15 mins followed by mouse a... |
Bioorg Med Chem Lett 30: (2020)
Article DOI: 10.1016/j.bmcl.2019.126886
BindingDB Entry DOI: 10.7270/Q26Q21RR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50217036
(CHEMBL74983)Show InChI InChI=1S/C14H8O2S3/c15-6-9-5-14(17-8-9)13-4-3-12(19-13)11-2-1-10(7-16)18-11/h1-8H | PDB
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| n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C |
Bioorg Med Chem Lett 9: 2279-82 (1999)
BindingDB Entry DOI: 10.7270/Q2MW2K90 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1 | PDB
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| n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Tokyo University of Agriculture
Curated by ChEMBL
| Assay Description
Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of ionomycin-stimulated beta-hexosaminidase release preincubated for 15 mins followed by... |
Bioorg Med Chem Lett 30: (2020)
Article DOI: 10.1016/j.bmcl.2019.126886
BindingDB Entry DOI: 10.7270/Q26Q21RR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1 | PDB
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| n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Tokyo University of Agriculture
Curated by ChEMBL
| Assay Description
Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of ionomycin-stimulated TNFalpha release preincubated for 15 mins followed by ionomycin ... |
Bioorg Med Chem Lett 30: (2020)
Article DOI: 10.1016/j.bmcl.2019.126886
BindingDB Entry DOI: 10.7270/Q26Q21RR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50213431
(CHEMBL84654)Show SMILES CCCCCCCCCCC#Cc1cccc(c1)[C@@H](O)[C@@H](N)CO |r| Show InChI InChI=1S/C21H33NO2/c1-2-3-4-5-6-7-8-9-10-11-13-18-14-12-15-19(16-18)21(24)20(22)17-23/h12,14-16,20-21,23-24H,2-10,17,22H2,1H3/t20-,21+/m0/s1 | PDB
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| | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50213427
(CHEMBL82271)Show SMILES CCCCCCCCCCC#Cc1ccc(s1)[C@@H](O)[C@@H](N)CO |r| Show InChI InChI=1S/C19H31NO2S/c1-2-3-4-5-6-7-8-9-10-11-12-16-13-14-18(23-16)19(22)17(20)15-21/h13-14,17,19,21-22H,2-10,15,20H2,1H3/t17-,19-/m0/s1 | PDB
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| | n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50217032
(CHEMBL76100)Show InChI InChI=1S/C13H10OS3/c14-7-9-6-13(16-8-9)12-4-3-11(17-12)10-2-1-5-15-10/h1-6,8,14H,7H2 | PDB
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| n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C |
Bioorg Med Chem Lett 9: 2279-82 (1999)
BindingDB Entry DOI: 10.7270/Q2MW2K90 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50213449
(CHEMBL82095)Show SMILES CCCCCCCCCCCC#Cc1ccc(s1)[C@@H](O)[C@@H](N)CO Show InChI InChI=1S/C20H33NO2S/c1-2-3-4-5-6-7-8-9-10-11-12-13-17-14-15-19(24-17)20(23)18(21)16-22/h14-15,18,20,22-23H,2-11,16,21H2,1H3/t18-,20-/m0/s1 | PDB
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| | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50213438
(CHEMBL83961)Show InChI InChI=1S/C21H37NO2/c1-2-3-4-5-6-7-8-9-10-11-13-18-14-12-15-19(16-18)21(24)20(22)17-23/h12,14-16,20-21,23-24H,2-11,13,17,22H2,1H3/t20-,21+/m0/s1 | PDB
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| | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50230709
(CHEMBL295954)Show InChI InChI=1S/C22H46NO2.BrH/c1-5-6-7-8-9-10-11-12-13-14-15-16-17-18-22(24-4)21-23(2,3)19-20-25-22;/h5-21H2,1-4H3;1H/q+1;/p-1 | PDB
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| n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C (PKC) purified from rat brain |
J Med Chem 36: 177-8 (1993)
BindingDB Entry DOI: 10.7270/Q2Z321VQ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50213426
(CHEMBL79293)Show SMILES CCCCCCCCCCCCCCCCc1cccc(n1)[C@@H](O)[C@@H](N)CO Show InChI InChI=1S/C24H44N2O2/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-17-21-18-16-19-23(26-21)24(28)22(25)20-27/h16,18-19,22,24,27-28H,2-15,17,20,25H2,1H3/t22-,24-/m0/s1 | PDB
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| | n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50213428
(CHEMBL309649)Show InChI InChI=1S/C18H29NO2S/c1-2-3-4-5-6-7-8-9-10-11-15-12-13-17(22-15)18(21)16(19)14-20/h12-13,16,18,20-21H,2-9,14,19H2,1H3/t16-,18-/m0/s1 | PDB
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| | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50217040
(CHEMBL73495)Show InChI InChI=1S/C13H8OS3/c14-7-9-6-13(16-8-9)12-4-3-11(17-12)10-2-1-5-15-10/h1-8H | PDB
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| n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C |
Bioorg Med Chem Lett 9: 2279-82 (1999)
BindingDB Entry DOI: 10.7270/Q2MW2K90 |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50213451
(CHEMBL86221)Show SMILES CCCCCCCCCC\C=C\c1csc(c1)[C@@H](O)[C@@H](N)CO Show InChI InChI=1S/C19H33NO2S/c1-2-3-4-5-6-7-8-9-10-11-12-16-13-18(23-15-16)19(22)17(20)14-21/h11-13,15,17,19,21-22H,2-10,14,20H2,1H3/b12-11+/t17-,19-/m0/s1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50230703
(CHEMBL296591)Show SMILES [Br-].CCCCCCCCCCCCCCCCCCC1(O)C[N+](C)(C)CCO1 Show InChI InChI=1S/C24H50NO2.BrH/c1-4-5-6-7-8-9-10-11-12-13-14-15-16-17-18-19-20-24(26)23-25(2,3)21-22-27-24;/h26H,4-23H2,1-3H3;1H/q+1;/p-1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C (PKC) purified from rat brain |
J Med Chem 36: 177-8 (1993)
BindingDB Entry DOI: 10.7270/Q2Z321VQ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM83205
((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)Show InChI InChI=1S/C18H37NO2/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-18(21)17(19)16-20/h14-15,17-18,20-21H,2-13,16,19H2,1H3/b15-14+/t17-,18+/m0/s1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| Purchase
MCE
KEGG
PC cid
PC sid
PDB
UniChem
Similars
| | n/a | n/a | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q21J9CZZ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50230702
(CHEMBL48695)Show InChI InChI=1S/C22H46NO2/c1-4-5-6-7-8-9-10-11-12-13-14-15-16-18-22(25)21-23(2,3)19-17-20-24/h24H,4-21H2,1-3H3/q+1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 6.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C (PKC) purified from rat brain |
J Med Chem 36: 177-8 (1993)
BindingDB Entry DOI: 10.7270/Q2Z321VQ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50230712
(CHEMBL52232)Show SMILES [Br-].CCCCCCCCCCCCCCCCCC1(O)C[N+](C)(C)CCO1 Show InChI InChI=1S/C23H48NO2.BrH/c1-4-5-6-7-8-9-10-11-12-13-14-15-16-17-18-19-23(25)22-24(2,3)20-21-26-23;/h25H,4-22H2,1-3H3;1H/q+1;/p-1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| n/a | n/a | 7.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C (PKC) purified from rat brain |
J Med Chem 36: 177-8 (1993)
BindingDB Entry DOI: 10.7270/Q2Z321VQ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50230714
(CHEMBL48551)Show InChI InChI=1S/C21H44NO2.BrH/c1-4-5-6-7-8-9-10-11-12-13-14-15-16-17-21(23)20-22(2,3)18-19-24-21;/h23H,4-20H2,1-3H3;1H/q+1;/p-1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| n/a | n/a | 7.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C (PKC) purified from rat brain |
J Med Chem 36: 177-8 (1993)
BindingDB Entry DOI: 10.7270/Q2Z321VQ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50230711
(CHEMBL441041)Show InChI InChI=1S/C20H42NO2.BrH/c1-4-5-6-7-8-9-10-11-12-13-14-15-16-20(22)19-21(2,3)17-18-23-20;/h22H,4-19H2,1-3H3;1H/q+1;/p-1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C (PKC) purified from rat brain |
J Med Chem 36: 177-8 (1993)
BindingDB Entry DOI: 10.7270/Q2Z321VQ |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Rattus norvegicus) | BDBM50230705
(CHEMBL49951)Show InChI InChI=1S/C22H46NO2.BrH/c1-4-5-6-7-8-9-10-11-12-13-14-15-16-17-18-22(24)21-23(2,3)19-20-25-22;/h24H,4-21H2,1-3H3;1H/q+1;/p-1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University
Curated by ChEMBL
| Assay Description
Inhibition of protein kinase C (PKC) purified from rat brain |
J Med Chem 36: 177-8 (1993)
BindingDB Entry DOI: 10.7270/Q2Z321VQ |
More data for this
Ligand-Target Pair | |
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