Found 3 hits of ec50 for UniProtKB: P51828 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Adenylate cyclase type 1/2/3/4/5/6/7/8/9
(Homo sapiens (Human)) | BDBM50004822
((R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine...)Show InChI InChI=1S/C16H17NO2/c18-15-8-12-6-7-17-10-14(13(12)9-16(15)19)11-4-2-1-3-5-11/h1-5,8-9,14,17-19H,6-7,10H2/t14-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| PubMed
| n/a | n/a | n/a | n/a | 71 | n/a | n/a | n/a | n/a |
University of Lund
Curated by ChEMBL
| Assay Description Compound was tested for the adenylate cyclase stimulation |
J Med Chem 35: 502-7 (1992)
BindingDB Entry DOI: 10.7270/Q2TH8N95 |
More data for this Ligand-Target Pair | |
Adenylate cyclase type 1/2/3/4/5/6/7/8/9
(Homo sapiens (Human)) | BDBM50004821
(2,3,4,5-Tetrahydro-1H-benzo[d]azepine-7,8-diol | C...)Show InChI InChI=1S/C10H13NO2/c12-9-5-7-1-3-11-4-2-8(7)6-10(9)13/h5-6,11-13H,1-4H2 | PDB
UniProtKB/SwissProt
antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Patents
Similars
| PubMed
| n/a | n/a | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a |
University of Lund
Curated by ChEMBL
| Assay Description Compound was tested for the adenylate cyclase stimulation |
J Med Chem 35: 502-7 (1992)
BindingDB Entry DOI: 10.7270/Q2TH8N95 |
More data for this Ligand-Target Pair | |
Adenylate cyclase type 1/2/3/4/5/6/7/8/9
(Homo sapiens (Human)) | BDBM50230364
(CHEMBL146629)Show InChI InChI=1S/C16H23NO2/c18-15-8-12-6-7-17-10-14(13(12)9-16(15)19)11-4-2-1-3-5-11/h8-9,11,14,17-19H,1-7,10H2/t14-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Lund
Curated by ChEMBL
| Assay Description Compound was tested for the adenylate cyclase stimulation |
J Med Chem 35: 502-7 (1992)
BindingDB Entry DOI: 10.7270/Q2TH8N95 |
More data for this Ligand-Target Pair | |