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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for UniProtKB: P19357   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Solute carrier family 2, facilitated glucose transporter member 4


(Rattus norvegicus)		BDBM50277370
PNG
(CHEMBL4171968)
Show SMILES COc1ccc(cc1)C(=O)N(Cc1ccncc1)Cc1cccc(OCCc2ccc(F)cc2)c1
Show InChI InChI=1S/C29H27FN2O3/c1-34-27-11-7-25(8-12-27)29(33)32(20-23-13-16-31-17-14-23)21-24-3-2-4-28(19-24)35-18-15-22-5-9-26(30)10-6-22/h2-14,16-17,19H,15,18,20-21H2,1H3
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 1.70E+3n/an/an/an/an/an/a



Emory University

Curated by ChEMBL


Assay Description
Antagonist activity at rat C-terminal 6His/Myc-tagged GLUT4 assessed as reduction in 2-[3H]deoxyglucose uptake measured after 6 mins

Eur J Med Chem 139: 573-586 (2017)


Article DOI: 10.1016/j.ejmech.2017.08.029
BindingDB Entry DOI: 10.7270/Q2NC63Q7
More data for this
Ligand-Target Pair