Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential cation channel, subfamily V, member 3 (Rattus norvegicus) | BDBM50285610 (CBV | CHEMBL4170268) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a |
University of Eastern Piedmont Curated by ChEMBL | Assay Description Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor... | J Nat Prod 81: 630-633 (2018) Article DOI: 10.1021/acs.jnatprod.7b00946 BindingDB Entry DOI: 10.7270/Q26D5WJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel, subfamily V, member 3 (Rattus norvegicus) | BDBM50061117 (6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol |...) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a |
University of Eastern Piedmont Curated by ChEMBL | Assay Description Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor... | J Nat Prod 81: 630-633 (2018) Article DOI: 10.1021/acs.jnatprod.7b00946 BindingDB Entry DOI: 10.7270/Q26D5WJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel, subfamily V, member 3 (Rattus norvegicus) | BDBM50463447 (CHEMBL4249046) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6.70E+3 | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Agonist activity at rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assay | Bioorg Med Chem 26: 4532-4536 (2018) Article DOI: 10.1016/j.bmc.2018.07.044 BindingDB Entry DOI: 10.7270/Q2M32ZFD | |||||||||||
More data for this Ligand-Target Pair |