Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Virulence sensor histidine kinase PhoQ (Salmonella typhimurium (strain LT2 / SGSC1412 / AT...) | BDBM50453878 (CHEMBL371380) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.38E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Williams College Curated by ChEMBL | Assay Description Inhibition of recombinant Salmonella typhimurium N-terminal His6-SUMO-tagged DHp-catalytic domain PhoQ (257 to 487 residues) autophosphorylation expr... | Bioorg Med Chem Lett 27: 5235-5244 (2017) Article DOI: 10.1016/j.bmcl.2017.10.036 BindingDB Entry DOI: 10.7270/Q20G3NQV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Virulence sensor histidine kinase PhoQ (Salmonella typhimurium (strain LT2 / SGSC1412 / AT...) | BDBM50453881 (CCT018159 | CHEBI:41656 | CHEMBL399530) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 2.61E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Williams College Curated by ChEMBL | Assay Description Inhibition of recombinant Salmonella typhimurium N-terminal His6-SUMO-tagged DHp-catalytic domain PhoQ (257 to 487 residues) autophosphorylation expr... | Bioorg Med Chem Lett 27: 5235-5244 (2017) Article DOI: 10.1016/j.bmcl.2017.10.036 BindingDB Entry DOI: 10.7270/Q20G3NQV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Virulence sensor histidine kinase PhoQ (Salmonella typhimurium (strain LT2 / SGSC1412 / AT...) | BDBM15364 (4-chloro-6-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.70E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Williams College Curated by ChEMBL | Assay Description Inhibition of recombinant Salmonella typhimurium N-terminal His6-SUMO-tagged DHp-catalytic domain PhoQ (257 to 487 residues) autophosphorylation expr... | Bioorg Med Chem Lett 27: 5235-5244 (2017) Article DOI: 10.1016/j.bmcl.2017.10.036 BindingDB Entry DOI: 10.7270/Q20G3NQV | |||||||||||
More data for this Ligand-Target Pair |