Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Virulence sensor histidine kinase PhoQ (Salmonella typhimurium (strain LT2 / SGSC1412 / AT...) | BDBM50453877 (CHEMBL4209514) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.91E+5 | n/a | n/a | n/a | n/a | n/a |
Williams College Curated by ChEMBL | Assay Description Displacement of TNP-ATP from recombinant Salmonella typhimurium GST-tagged DHp-catalytic domain PhoQ (332 to 487 residues) expressed in Escherichia c... | Bioorg Med Chem Lett 27: 5235-5244 (2017) Article DOI: 10.1016/j.bmcl.2017.10.036 BindingDB Entry DOI: 10.7270/Q20G3NQV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Virulence sensor histidine kinase PhoQ (Salmonella typhimurium (strain LT2 / SGSC1412 / AT...) | BDBM227589 (Radicicol) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 7.15E+5 | n/a | n/a | n/a | n/a | n/a |
Williams College Curated by ChEMBL | Assay Description Binding affinity to recombinant Salmonella typhimurium 15N-labeled PhoQ catalytic domain (332 to 487 residues) expressed in Escherichia coli XA90 ass... | Bioorg Med Chem Lett 27: 5235-5244 (2017) Article DOI: 10.1016/j.bmcl.2017.10.036 BindingDB Entry DOI: 10.7270/Q20G3NQV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |