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Compile Data Set for Download or QSAR

Found 1 hit of ic50 data for polymerid = 50007795   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Tolloid-like protein 1


(Homo sapiens)		BDBM50458762
PNG
(CHEMBL4207308)
Show SMILES CCCCC[C@H]([C@@H](CC)N(O)C=O)C(=O)NCNC(=O)c1ccc(o1)-c1ccccc1 |r|
Show InChI InChI=1S/C23H31N3O5/c1-3-5-7-12-18(19(4-2)26(30)16-27)22(28)24-15-25-23(29)21-14-13-20(31-21)17-10-8-6-9-11-17/h6,8-11,13-14,16,18-19,30H,3-5,7,12,15H2,1-2H3,(H,24,28)(H,25,29)/t18-,19-/m1/s1
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem
Article
PubMed
n/an/a 100n/an/an/an/an/an/a



GlaxoSmithKline Pharmaceuticals

Curated by ChEMBL


Assay Description
Inhibition of PI3Kgamma (2 to 1102) (unknown origin) using diC8-PIP2 as substrate preincubated for 30 mins followed by substrate addition measured af...

ACS Med Chem Lett 9: 736-740 (2018)


Article DOI: 10.1021/acsmedchemlett.8b00173
BindingDB Entry DOI: 10.7270/Q2X35127
More data for this
Ligand-Target Pair