BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit of kd for UniProtKB: P00533   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Epidermal growth factor receptor [1-746,748-748,750-1210,A750P]


(Homo sapiens (Human))		BDBM373711
PNG
(US10246444, Example 40)
Show SMILES CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)CC1CCSS1
Show InChI InChI=1S/C30H26ClFN4O3S2/c1-2-38-28-14-25-23(13-26(28)36-29(37)12-22-8-9-40-41-22)30(19(15-33)16-34-25)35-21-6-7-27(24(31)11-21)39-17-18-4-3-5-20(32)10-18/h3-7,10-11,13-14,16,22H,2,8-9,12,17H2,1H3,(H,34,35)(H,36,37)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/a 50n/an/an/an/an/a



St. Jude Research Hospital



Assay Description
KINOMEscan is based on a competition binding assay that quantitatively measures the ability of a compound to compete with an immobilized, active-site...

J Med Chem 50: 1876-85 (2007)


BindingDB Entry DOI: 10.7270/Q2NC63HJ
More data for this
Ligand-Target Pair