Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DNA-directed RNA polymerase subunit alpha () | BDBM466524 (US10800725, Compound 12) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466521 (US10800725, Compound 9) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 840 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466519 (US10800725, Compound 7) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466522 (US10800725, Compound 10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466520 (US10800725, Compound 8) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466515 (US10800725, Compound 3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466517 (US10800725, Compound 5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466526 (US10800725, Compound 14) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466523 (US10800725, Compound 11) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466518 (US10800725, Compound 6) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466516 (US10800725, Compound 4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466525 (US10800725, Compound 13) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466513 (US10800725, Compound 1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466514 (US10800725, Compound 2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466507 (US10800725, Compound 15) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466512 (US10800725, Compound 20) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466511 (US10800725, Compound 19) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466510 (US10800725, Compound 18) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466509 (US10800725, Compound 17) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA-directed RNA polymerase subunit alpha () | BDBM466508 (US10800725, Compound 16) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA US Patent | Assay Description Fluorescence-detected RNA polymerase assays with S. aureus RNA polymerase were performed as in Example 21.1, using reaction mixtures containing (20 &... | US Patent US10800725 (2020) BindingDB Entry DOI: 10.7270/Q2GB274V | |||||||||||
More data for this Ligand-Target Pair |