Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium/potassium-transporting ATPase subunit alpha-1 (Homo sapiens (Human)) | BDBM46355 (DIGOXIN | MLS000069819 | SMR000059217 | US10668094...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal de S£o Jo£o Del Rei Curated by ChEMBL | Assay Description Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric method | Bioorg Med Chem 23: 4397-404 (2015) Article DOI: 10.1016/j.bmc.2015.06.028 BindingDB Entry DOI: 10.7270/Q2MG7R8C | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Sodium/potassium-transporting ATPase subunit alpha-1 (Homo sapiens (Human)) | BDBM50096255 (CHEMBL3594278) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal de S£o Jo£o Del Rei Curated by ChEMBL | Assay Description Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric method | Bioorg Med Chem 23: 4397-404 (2015) Article DOI: 10.1016/j.bmc.2015.06.028 BindingDB Entry DOI: 10.7270/Q2MG7R8C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium/potassium-transporting ATPase subunit alpha-1 (Homo sapiens (Human)) | BDBM50096254 (CHEMBL3594276) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal de S£o Jo£o Del Rei Curated by ChEMBL | Assay Description Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric method | Bioorg Med Chem 23: 4397-404 (2015) Article DOI: 10.1016/j.bmc.2015.06.028 BindingDB Entry DOI: 10.7270/Q2MG7R8C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium/potassium-transporting ATPase subunit alpha-1 (Homo sapiens (Human)) | BDBM50096256 (CHEMBL3594279) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal de S£o Jo£o Del Rei Curated by ChEMBL | Assay Description Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric method | Bioorg Med Chem 23: 4397-404 (2015) Article DOI: 10.1016/j.bmc.2015.06.028 BindingDB Entry DOI: 10.7270/Q2MG7R8C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium/potassium-transporting ATPase subunit alpha-1 (Homo sapiens (Human)) | BDBM50096257 (CHEMBL3594280) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal de S£o Jo£o Del Rei Curated by ChEMBL | Assay Description Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric method | Bioorg Med Chem 23: 4397-404 (2015) Article DOI: 10.1016/j.bmc.2015.06.028 BindingDB Entry DOI: 10.7270/Q2MG7R8C | |||||||||||
More data for this Ligand-Target Pair |