Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ras guanyl-releasing protein 3 (Homo sapiens (Human)) | BDBM50106245 (2-{4-hydroxy-3-hydroxymethyl-2-(3-hydroxypropyl)-4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Michigan Cancer Center Curated by ChEMBL | Assay Description Binding affinity for RasGPR3, guanine nucleotide exchange factor | J Med Chem 44: 3872-80 (2001) BindingDB Entry DOI: 10.7270/Q2Z037F5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras guanyl-releasing protein 3 (Homo sapiens (Human)) | BDBM50106244 (6-[9-[1-formyl-(Z)-ethylidene]-1,6-dihydroxy-10-(3...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Michigan Cancer Center Curated by ChEMBL | Assay Description Binding affinity for RasGPR3, guanine nucleotide exchange factor | J Med Chem 44: 3872-80 (2001) BindingDB Entry DOI: 10.7270/Q2Z037F5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Homo sapiens (Human)) | BDBM50106245 (2-{4-hydroxy-3-hydroxymethyl-2-(3-hydroxypropyl)-4...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 76 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Michigan Cancer Center Curated by ChEMBL | Assay Description Binding affinity for PKC alpha (C1b domain) | J Med Chem 44: 3872-80 (2001) BindingDB Entry DOI: 10.7270/Q2Z037F5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Homo sapiens (Human)) | BDBM50106244 (6-[9-[1-formyl-(Z)-ethylidene]-1,6-dihydroxy-10-(3...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 84 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Michigan Cancer Center Curated by ChEMBL | Assay Description Binding affinity for PKC alpha (C1b domain) | J Med Chem 44: 3872-80 (2001) BindingDB Entry DOI: 10.7270/Q2Z037F5 | |||||||||||
More data for this Ligand-Target Pair |