BindingDB PrimarySearch

Found 12 hits Enz. Inhib. hit(s) with all data for entry = 50034127
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein kinase C delta type (Homo sapiens (Human))	BDBM50163748 ((E)-3,5-Bis[beta-(4-Hydroxy-3-methoxyphenyl)-ethen...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.50E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50357492 (CHEMBL1914609) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.16E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50163745 (4,40-(1E,10E)-2,20-(Isoxazole-3,5-diyl)bis(ethene-...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.16E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50357493 (CHEMBL1914610) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.52E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM50163748 ((E)-3,5-Bis[beta-(4-Hydroxy-3-methoxyphenyl)-ethen...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.88E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCepsilon C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C theta type (Homo sapiens (Human))	BDBM50357493 (CHEMBL1914610) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	7.14E+3	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCtheta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM50163745 (4,40-(1E,10E)-2,20-(Isoxazole-3,5-diyl)bis(ethene-...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.18E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCepsilon C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM50357493 (CHEMBL1914610) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.34E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCepsilon C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C theta type (Homo sapiens (Human))	BDBM50163748 ((E)-3,5-Bis[beta-(4-Hydroxy-3-methoxyphenyl)-ethen...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	7.25E+3	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCtheta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C theta type (Homo sapiens (Human))	BDBM50357492 (CHEMBL1914609) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.58E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCtheta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C theta type (Homo sapiens (Human))	BDBM50163745 (4,40-(1E,10E)-2,20-(Isoxazole-3,5-diyl)bis(ethene-...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	3.16E+3	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCtheta C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM50357492 (CHEMBL1914609) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.61E+4	n/a	n/a	n/a	n/a
University of Houston Curated by ChEMBL					Assay Description Binding affinity to PKCepsilon C1B subdomain after 1 hr by fluorescence quenching analysis				Bioorg Med Chem 19: 6196-202 (2011) Article DOI: 10.1016/j.bmc.2011.09.011 BindingDB Entry DOI: 10.7270/Q2BK1CST
University of Houston Curated by ChEMBL					More data for this Ligand-Target Pair