Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tubulin beta chain (Sus scrofa) | BDBM50483304 (11-Epi-Tubulysin D) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyorin Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by microtubule assembly assay | Bioorg Med Chem Lett 21: 431-4 (2011) Article DOI: 10.1016/j.bmcl.2010.10.118 BindingDB Entry DOI: 10.7270/Q21J9DMW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin beta chain (Sus scrofa) | BDBM50012278 ((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyorin Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by microtubule assembly assay | Bioorg Med Chem Lett 21: 431-4 (2011) Article DOI: 10.1016/j.bmcl.2010.10.118 BindingDB Entry DOI: 10.7270/Q21J9DMW | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Tubulin beta chain (Sus scrofa) | BDBM50483305 (13-Epi-Tubulysin D) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyorin Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by microtubule assembly assay | Bioorg Med Chem Lett 21: 431-4 (2011) Article DOI: 10.1016/j.bmcl.2010.10.118 BindingDB Entry DOI: 10.7270/Q21J9DMW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin beta chain (Sus scrofa) | BDBM50483306 (CHEBI:80036 | Tubulysin D) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyorin Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by microtubule assembly assay | Bioorg Med Chem Lett 21: 431-4 (2011) Article DOI: 10.1016/j.bmcl.2010.10.118 BindingDB Entry DOI: 10.7270/Q21J9DMW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin beta chain (Sus scrofa) | BDBM50483307 (CHEMBL1643767) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyorin Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by microtubule assembly assay | Bioorg Med Chem Lett 21: 431-4 (2011) Article DOI: 10.1016/j.bmcl.2010.10.118 BindingDB Entry DOI: 10.7270/Q21J9DMW | |||||||||||
More data for this Ligand-Target Pair |