Found 35 hits Enz. Inhib. hit(s) with all data for entry = 50014580 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577608
(CHEMBL4847166) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577605
(CHEMBL4876917) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577604
(CHEMBL4855258) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577611
(CHEMBL4848633) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577613
(CHEMBL4857804) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity in... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577613
(CHEMBL4857804) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577610
(CHEMBL4877438) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577615
(CHEMBL4867055) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577605
(CHEMBL4876917) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 monomer response element NBRE expressed in HEK293T cells co-expressing firefly luciferase assessed... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577609
(CHEMBL4853371) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577597
(CHEMBL4854333) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577612
(CHEMBL4860059) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577613
(CHEMBL4857804) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 monomer response element NBRE expressed in HEK293T cells co-expressing firefly luciferase assessed... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577614
(CHEMBL4848553) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577606
(CHEMBL4867759) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577603
(CHEMBL4877114) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577599
(CHEMBL4864410) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577594
(CHEMBL4863910) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577600
(CHEMBL4877456) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577602
(CHEMBL4863919) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577595
(CHEMBL4860942) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577613
(CHEMBL4857804) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at human Nurr1 LBD assessed as displacement of NCoR2 from Nurr1 after 2 hrs by HTRF assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577607
(CHEMBL4863805) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577601
(CHEMBL4850618) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577592
(CHEMBL4862487) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 3.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577598
(CHEMBL4852316) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50250885
(CHEBI:65019 | CHEMBL2270066)Show InChI InChI=1S/C10H9NO2/c1-13-10(12)8-6-11-9-5-3-2-4-7(8)9/h2-6,11H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid PDB UniChem
Similars
| Article PubMed
| n/a | n/a | 4.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577591
(CHEMBL4857839) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 5.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577593
(CHEMBL4855705) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577613
(CHEMBL4857804) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 5.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at human Nurr1 LBD assessed as displacement of NCoR1 from Nurr1 after 2 hrs by HTRF assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577596
(CHEMBL4862520) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 5.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Inverse agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50041457
(4-[(7-chloroquinolin-4-yl)amino]-2-[(diethylamino)...)Show InChI InChI=1S/C20H22ClN3O/c1-3-24(4-2)13-14-11-16(6-8-20(14)25)23-18-9-10-22-19-12-15(21)5-7-17(18)19/h5-12,25H,3-4,13H2,1-2H3,(H,22,23) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 8.20E+4 | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity in presenc... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577617
(CHEMBL4872383) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by hybrid ... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50577616
(CHEMBL4860845) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | n/a | n/a | 8.10E+4 | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by hybrid ... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human)) | BDBM50041457
(4-[(7-chloroquinolin-4-yl)amino]-2-[(diethylamino)...)Show InChI InChI=1S/C20H22ClN3O/c1-3-24(4-2)13-14-11-16(6-8-20(14)25)23-18-9-10-22-19-12-15(21)5-7-17(18)19/h5-12,25H,3-4,13H2,1-2H3,(H,22,23) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 4.10E+4 | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity by hybrid ... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.1c01077 BindingDB Entry DOI: 10.7270/Q27W6H24 |
More data for this Ligand-Target Pair | |