Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50004000 ((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110325 (CHEMBL3605423) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.71E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110253 (CHEMBL3605418) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110316 (CHEMBL3605434) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.24E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110252 (CHEMBL3605419) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.33E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110255 (CHEMBL3605316) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.38E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110317 (CHEMBL3605433) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.61E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110324 (CHEMBL3605424) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.88E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110314 (CHEMBL3605437) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.52E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110322 (CHEMBL3605426) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.61E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110320 (CHEMBL3605430) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110278 (CHEMBL3605309) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110257 (CHEMBL3605314) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.88E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110326 (CHEMBL3605422) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.13E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110318 (CHEMBL3605432) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110323 (CHEMBL3605425) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110261 (CHEMBL3605313) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110277 (CHEMBL3605310) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110279 (CHEMBL3605308) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110319 (CHEMBL3605431) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110321 (CHEMBL3605428) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Homo sapiens (Human)) | BDBM50110315 (CHEMBL3605436) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Punjab Curated by ChEMBL | Assay Description Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 30 mins before substrate addition measured after 30 ... | Bioorg Med Chem 23: 6014-24 (2015) Article DOI: 10.1016/j.bmc.2015.06.051 BindingDB Entry DOI: 10.7270/Q2TT4SQS | |||||||||||
More data for this Ligand-Target Pair |