Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50378798 (CYTOSPORONE B) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 0.278 | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Agonist activity at nuclear orphan receptor Nur77 expressed in human BGC823 cells co-transfected with fused GAL4-Nur77 assessed as transactivation af... | Nat Chem Biol 4: 548-56 (2008) Article DOI: 10.1038/nchembio.106 BindingDB Entry DOI: 10.7270/Q2959JHW | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |