Found 233 hits Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase 10' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM93207
(Kinase inhibitor, 5)Show SMILES Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccc2nc(Nc3ccc(OCCN)cc3)ncc2c1 Show InChI InChI=1S/C31H26F3N5O2/c1-19-5-7-25(37-29(40)21-3-2-4-23(16-21)31(32,33)34)17-27(19)20-6-12-28-22(15-20)18-36-30(39-28)38-24-8-10-26(11-9-24)41-14-13-35/h2-12,15-18H,13-14,35H2,1H3,(H,37,40)(H,36,38,39) | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | <10 | n/a | n/a | n/a | n/a | 7.5 | 25 |
University of Washington
| Assay Description Fluorescence assay used for determination of catch and release efficiency. |
ACS Chem Biol 8: 691-9 (2013)
Article DOI: 10.1021/cb300623a BindingDB Entry DOI: 10.7270/Q20R9N1X |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM93207
(Kinase inhibitor, 5)Show SMILES Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccc2nc(Nc3ccc(OCCN)cc3)ncc2c1 Show InChI InChI=1S/C31H26F3N5O2/c1-19-5-7-25(37-29(40)21-3-2-4-23(16-21)31(32,33)34)17-27(19)20-6-12-28-22(15-20)18-36-30(39-28)38-24-8-10-26(11-9-24)41-14-13-35/h2-12,15-18H,13-14,35H2,1H3,(H,37,40)(H,36,38,39) | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | <20 | n/a | n/a | n/a | n/a | 7.5 | 25 |
University of Washington
| Assay Description Fluorescence assay used for determination of catch and release efficiency. |
ACS Chem Biol 8: 691-9 (2013)
Article DOI: 10.1021/cb300623a BindingDB Entry DOI: 10.7270/Q20R9N1X |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577328
(CHEMBL4875188)Show SMILES COc1ccccc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577368
(CHEMBL4878325)Show SMILES COc1cc(Br)ccc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O |c:10| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8226
(3-[(3-chlorophenyl)amino]-4-(2-methoxyphenyl)-2,5-...)Show SMILES COc1ccccc1C1=C(Nc2cccc(Cl)c2)C(=O)NC1=O |c:9| Show InChI InChI=1S/C17H13ClN2O3/c1-23-13-8-3-2-7-12(13)14-15(17(22)20-16(14)21)19-11-6-4-5-10(18)9-11/h2-9H,1H3,(H2,19,20,21,22) | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
Similars
| Article PubMed
| 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577340
(CHEMBL4877889)Show SMILES COc1ccccc1C1=C(Nc2cccc3ccccc23)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 47 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577369
(CHEMBL4856751)Show SMILES COc1ccc(Br)cc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O |c:10| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 61 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8244
(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(2-methoxyph...)Show SMILES COc1ccccc1C1=C(Nc2ccc(O)c(Cl)c2)C(=O)NC1=O |c:9| Show InChI InChI=1S/C17H13ClN2O4/c1-24-13-5-3-2-4-10(13)14-15(17(23)20-16(14)22)19-9-6-7-12(21)11(18)8-9/h2-8,21H,1H3,(H2,19,20,22,23) | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 73 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577318
(CHEMBL4855513)Show SMILES COc1ccccc1C1=C(Nc2cccc(F)c2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 76 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577338
(CHEMBL4869745)Show SMILES COc1ccccc1C1=C(Nc2ccc3OCOc3c2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 84 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577366
(CHEMBL4867952)Show SMILES COc1cc(NC(=O)C(C)C)ccc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O |c:15| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577308
(CHEMBL4857159)Show SMILES COc1ccccc1C1=C(Nc2cccc(SC)c2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577350
(CHEMBL4868821)Show SMILES COc1ccccc1C1=C(Nc2ccc3ncccc3c2)C(=O)NC1=O |c:9| | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577331
(CHEMBL4877101)Show SMILES O=C1NC(=O)C(=C1Nc1cccc(c1)C#N)c1cccc2ccccc12 |c:5| | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577334
(CHEMBL4852101)Show SMILES COc1ccc(NC2=C(C(=O)NC2=O)c2ccccc2OC)cc1 |t:7| | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8275
(3-(2-methoxyphenyl)-4-{[4-(methylsulfanyl)phenyl]a...)Show SMILES COc1ccccc1C1=C(Nc2ccc(SC)cc2)C(=O)NC1=O |c:9| Show InChI InChI=1S/C18H16N2O3S/c1-23-14-6-4-3-5-13(14)15-16(18(22)20-17(15)21)19-11-7-9-12(24-2)10-8-11/h3-10H,1-2H3,(H2,19,20,21,22) | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8243
(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(2-chlorophe...)Show SMILES Oc1ccc(NC2=C(C(=O)NC2=O)c2ccccc2Cl)cc1Cl |t:6| Show InChI InChI=1S/C16H10Cl2N2O3/c17-10-4-2-1-3-9(10)13-14(16(23)20-15(13)22)19-8-5-6-12(21)11(18)7-8/h1-7,21H,(H2,19,20,22,23) | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577333
(CHEMBL4847820)Show SMILES COc1cccc(NC2=C(C(=O)NC2=O)c2ccccc2OC)c1 |t:8| | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577315
(CHEMBL160338)Show SMILES COc1ccccc1C1=C(Nc2ccc(O)cc2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577314
(CHEMBL347702)Show SMILES Oc1ccc(NC2=C(C(=O)NC2=O)c2ccccc2Cl)cc1 |t:6| | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8225
(3-(2-chlorophenyl)-4-[(3-chlorophenyl)amino]-2,5-d...)Show SMILES Clc1cccc(NC2=C(C(=O)NC2=O)c2ccccc2Cl)c1 |t:7| Show InChI InChI=1S/C16H10Cl2N2O2/c17-9-4-3-5-10(8-9)19-14-13(15(21)20-16(14)22)11-6-1-2-7-12(11)18/h1-8H,(H2,19,20,21,22) | PDB MMDB
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UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577354
(CHEMBL4869281)Show SMILES COc1ccc(cc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O)-c1ccccc1 |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 320 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577365
(CHEMBL4845800)Show SMILES COc1cc(ccc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O)-c1ccc(Cl)nc1Cl |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 320 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577341
(CHEMBL4851482)Show SMILES COc1ccccc1C1=C(Nc2ccc(cc2)-c2ccccc2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 320 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577320
(CHEMBL4847807)Show SMILES COc1ccccc1C1=C(Nc2cccc(c2)C(F)(F)F)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577307
(CHEMBL4858023)Show SMILES CSc1cccc(NC2=C(C(=O)NC2=O)c2ccccc2Cl)c1 |t:8| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577327
(CHEMBL4848202)Show SMILES Clc1ccccc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O |c:8| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577317
(CHEMBL4878748)Show SMILES Fc1cccc(NC2=C(C(=O)NC2=O)c2ccccc2Cl)c1 |t:7| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577346
(CHEMBL4863077)Show SMILES COc1ccccc1C1=C(Nc2ccc(cc2)-c2ccsc2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577363
(CHEMBL4852451)Show SMILES COc1cc(ccc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O)-c1cccnc1 |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 440 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577339
(CHEMBL4854271)Show SMILES COc1ccccc1C1=C(Nc2ccc(cc2)N2CCOCC2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577337
(CHEMBL4848740)Show SMILES COc1cc(NC2=C(C(=O)NC2=O)c2ccccc2OC)cc(OC)c1 |t:6| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 480 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8234
(3-[(3-hydroxyphenyl)amino]-4-(2-methoxyphenyl)-2,5...)Show SMILES COc1ccccc1C1=C(Nc2cccc(O)c2)C(=O)NC1=O |c:9| Show InChI InChI=1S/C17H14N2O4/c1-23-13-8-3-2-7-12(13)14-15(17(22)19-16(14)21)18-10-5-4-6-11(20)9-10/h2-9,20H,1H3,(H2,18,19,21,22) | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 480 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577361
(CHEMBL4875006)Show SMILES COc1cc(ccc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O)-c1ccsc1 |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8233
(3-(2-chlorophenyl)-4-[(3-hydroxyphenyl)amino]-2,5-...)Show SMILES Oc1cccc(NC2=C(C(=O)NC2=O)c2ccccc2Cl)c1 |t:7| Show InChI InChI=1S/C16H11ClN2O3/c17-12-7-2-1-6-11(12)13-14(16(22)19-15(13)21)18-9-4-3-5-10(20)8-9/h1-8,20H,(H2,18,19,21,22) | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 560 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8219
(3-(2-chlorophenyl)-4-(phenylamino)-2,5-dihydro-1H-...)Show InChI InChI=1S/C16H11ClN2O2/c17-12-9-5-4-8-11(12)13-14(16(21)19-15(13)20)18-10-6-2-1-3-7-10/h1-9H,(H2,18,19,20,21) | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 560 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8251
(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-(2-metho...)Show SMILES COc1ccccc1C1=C(Nc2cc(Cl)c(O)c(Cl)c2)C(=O)NC1=O |c:9| Show InChI InChI=1S/C17H12Cl2N2O4/c1-25-12-5-3-2-4-9(12)13-14(17(24)21-16(13)23)20-8-6-10(18)15(22)11(19)7-8/h2-7,22H,1H3,(H2,20,21,23,24) | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 590 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577343
(CHEMBL4876254)Show SMILES COc1ccccc1C1=C(Nc2ccc(cc2)C(=O)c2ccccc2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid PDB UniChem
| PDB Article PubMed
| 600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | 3D Structure (crystal) |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577322
(CHEMBL4851803)Show SMILES Oc1ccc(NC2=C(C(=O)NC2=O)c2ccccc2C(F)(F)F)cc1Cl |t:6| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 610 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577311
(CHEMBL4877795)Show SMILES COc1ccccc1C1=C(Nc2cccc(c2)S(C)(=O)=O)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577345
(CHEMBL4855633)Show SMILES COc1ccccc1C1=C(Nc2cccc(c2)-c2ccsc2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 640 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577306
(CHEMBL4860051)Show SMILES CSc1cccc(NC2=C(C(=O)NC2=O)c2ccccc2C(F)(F)F)c1 |t:8| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 730 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8274
(3-(2-chlorophenyl)-4-{[4-(methylsulfanyl)phenyl]am...)Show SMILES CSc1ccc(NC2=C(C(=O)NC2=O)c2ccccc2Cl)cc1 |t:7| Show InChI InChI=1S/C17H13ClN2O2S/c1-23-11-8-6-10(7-9-11)19-15-14(16(21)20-17(15)22)12-4-2-3-5-13(12)18/h2-9H,1H3,(H2,19,20,21,22) | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 760 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577349
(CHEMBL4859423)Show SMILES COc1ccccc1C1=C(Nc2ccc(OCc3ccccc3)c(Cl)c2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 790 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM8228
(3-[(3-chlorophenyl)amino]-4-(3-methoxyphenyl)-2,5-...)Show SMILES COc1cccc(c1)C1=C(Nc2cccc(Cl)c2)C(=O)NC1=O |c:9| Show InChI InChI=1S/C17H13ClN2O3/c1-23-13-7-2-4-10(8-13)14-15(17(22)20-16(14)21)19-12-6-3-5-11(18)9-12/h2-9H,1H3,(H2,19,20,21,22) | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| Article PubMed
| 950 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577321
(CHEMBL4848852)Show SMILES FC(F)(F)c1ccccc1C1=C(Nc2cccc(Cl)c2)C(=O)NC1=O |c:11| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 960 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577362
(CHEMBL4870533)Show SMILES COc1ccc(cc1C1=C(Nc2cccc(c2)C#N)C(=O)NC1=O)-c1ccsc1 |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577336
(CHEMBL4876004)Show SMILES COc1ccc(NC2=C(C(=O)NC2=O)c2ccccc2OC)cc1OC |t:7| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577344
(CHEMBL4873631)Show SMILES COc1ccccc1C1=C(Nc2ccc(Nc3ccccc3)cc2)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |
Serine/threonine-protein kinase 10
(Homo sapiens (Human)) | BDBM50577305
(CHEMBL4878043)Show SMILES COc1ccccc1C1=C(Nc2ccccc2SC)C(=O)NC1=O |c:9| | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Binding affinity human STK10 by binding displacement assay |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01579 BindingDB Entry DOI: 10.7270/Q2ST7TPK |
More data for this Ligand-Target Pair | |