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Patent code US9409892

Compile Data Set for Download or QSAR

Found 368 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240906
PNG
(US9409892, 1)
Show SMILES OC(=O)CCNC(=O)c1ncc2cc(Oc3ccccc3)ccc2c1O
Show InChI InChI=1S/C19H16N2O5/c22-16(23)8-9-20-19(25)17-18(24)15-7-6-14(10-12(15)11-21-17)26-13-4-2-1-3-5-13/h1-7,10-11,24H,8-9H2,(H,20,25)(H,22,23)
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n/an/a 920n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240911
PNG
(US9409892, 6)
Show SMILES CC(C)(CC(O)=O)NC(=O)c1ncc2cc(Oc3ccccc3)ccc2c1O
Show InChI InChI=1S/C21H20N2O5/c1-21(2,11-17(24)25)23-20(27)18-19(26)16-9-8-15(10-13(16)12-22-18)28-14-6-4-3-5-7-14/h3-10,12,26H,11H2,1-2H3,(H,23,27)(H,24,25)
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n/an/a 8.19E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240916
PNG
(US9409892, 11)
Show SMILES CC(CC(O)=O)NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O
Show InChI InChI=1S/C21H17N3O5/c1-12(9-18(25)26)23-21(28)19-20(27)15-8-7-14(10-16(15)17(11-22)24-19)29-13-5-3-2-4-6-13/h2-8,10,12,27H,9H2,1H3,(H,23,28)(H,25,26)
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n/an/a 1.37E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240917
PNG
(US9409892, 12)
Show SMILES OC(=O)C1(CNC(=O)c2nc(C#N)c3cc(Oc4ccccc4)ccc3c2O)CC1
Show InChI InChI=1S/C22H17N3O5/c23-11-17-16-10-14(30-13-4-2-1-3-5-13)6-7-15(16)19(26)18(25-17)20(27)24-12-22(8-9-22)21(28)29/h1-7,10,26H,8-9,12H2,(H,24,27)(H,28,29)
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n/an/a 170n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240918
PNG
(US9409892, 13)
Show SMILES OC(=O)C1(CNC(=O)c2ncc3cc(Oc4ccccc4)ccc3c2O)CCC1
Show InChI InChI=1S/C22H20N2O5/c25-19-17-8-7-16(29-15-5-2-1-3-6-15)11-14(17)12-23-18(19)20(26)24-13-22(21(27)28)9-4-10-22/h1-3,5-8,11-12,25H,4,9-10,13H2,(H,24,26)(H,27,28)
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n/an/a 5.51E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240932
PNG
(US9409892, 27)
Show SMILES CC(C)(CNC(=O)c1nc(C#N)c2cc(Oc3cccnc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C21H18N4O5/c1-21(2,20(28)29)11-24-19(27)17-18(26)14-6-5-12(8-15(14)16(9-22)25-17)30-13-4-3-7-23-10-13/h3-8,10,26H,11H2,1-2H3,(H,24,27)(H,28,29)
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n/an/a 3.27E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240950
PNG
(US9409892, 45)
Show SMILES N[C@@H](CCNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)C(O)=O |r|
Show InChI InChI=1S/C21H18N4O5/c22-11-17-15-10-13(30-12-4-2-1-3-5-12)6-7-14(15)19(26)18(25-17)20(27)24-9-8-16(23)21(28)29/h1-7,10,16,26H,8-9,23H2,(H,24,27)(H,28,29)/t16-/m0/s1
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n/an/a 1.41E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241062
PNG
(US9409892, 157)
Show SMILES CC(C)(CNC(=O)c1c(O)c2ccc(Oc3ccccc3)cc2c(C#N)[n+]1[O-])C(O)=O
Show InChI InChI=1S/C22H19N3O6/c1-22(2,21(28)29)12-24-20(27)18-19(26)15-9-8-14(31-13-6-4-3-5-7-13)10-16(15)17(11-23)25(18)30/h3-10,26H,12H2,1-2H3,(H,24,27)(H,28,29)
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n/an/a 1.36E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241067
PNG
(US9409892, 162)
Show SMILES CC(C)(CNC(=O)c1nc(C#N)c2cc(NC(=O)NCc3ccccc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C24H23N5O5/c1-24(2,22(32)33)13-27-21(31)19-20(30)16-9-8-15(10-17(16)18(11-25)29-19)28-23(34)26-12-14-6-4-3-5-7-14/h3-10,30H,12-13H2,1-2H3,(H,27,31)(H,32,33)(H2,26,28,34)
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n/an/a 2.35E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241072
PNG
(US9409892, 167)
Show SMILES OC(=O)C(CNC(=O)c1ncc2cc(Oc3ccccc3)ccc2c1O)C1CC1
Show InChI InChI=1S/C22H20N2O5/c25-20-17-9-8-16(29-15-4-2-1-3-5-15)10-14(17)11-23-19(20)21(26)24-12-18(22(27)28)13-6-7-13/h1-5,8-11,13,18,25H,6-7,12H2,(H,24,26)(H,27,28)
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n/an/a 9.57E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241086
PNG
(US9409892, 181)
Show SMILES OC(=O)C(CNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)c1ccc(F)cc1
Show InChI InChI=1S/C26H18FN3O5/c27-16-8-6-15(7-9-16)21(26(33)34)14-29-25(32)23-24(31)19-11-10-18(12-20(19)22(13-28)30-23)35-17-4-2-1-3-5-17/h1-12,21,31H,14H2,(H,29,32)(H,33,34)
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n/an/a 1.45E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240916
PNG
(US9409892, 11)
Show SMILES CC(CC(O)=O)NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O
Show InChI InChI=1S/C21H17N3O5/c1-12(9-18(25)26)23-21(28)19-20(27)15-8-7-14(10-16(15)17(11-22)24-19)29-13-5-3-2-4-6-13/h2-8,10,12,27H,9H2,1H3,(H,23,28)(H,25,26)
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n/an/a 5.66E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240925
PNG
(US9409892, 20)
Show SMILES COc1ccc(Oc2ccc3c(O)c(nc(C#N)c3c2)C(=O)NCC(C)(C)C(O)=O)cc1
Show InChI InChI=1S/C23H21N3O6/c1-23(2,22(29)30)12-25-21(28)19-20(27)16-9-8-15(10-17(16)18(11-24)26-19)32-14-6-4-13(31-3)5-7-14/h4-10,27H,12H2,1-3H3,(H,25,28)(H,29,30)
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n/an/a 5.22E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240930
PNG
(US9409892, 25)
Show SMILES OC(=O)CCNC(=O)c1ncc2cc(Oc3ccccn3)ccc2c1O
Show InChI InChI=1S/C18H15N3O5/c22-15(23)6-8-20-18(25)16-17(24)13-5-4-12(9-11(13)10-21-16)26-14-3-1-2-7-19-14/h1-5,7,9-10,24H,6,8H2,(H,20,25)(H,22,23)
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n/an/a 4.46E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240942
PNG
(US9409892, 37)
Show SMILES OC[C@@H](CC(O)=O)NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O |r|
Show InChI InChI=1S/C21H17N3O6/c22-10-17-16-9-14(30-13-4-2-1-3-5-13)6-7-15(16)20(28)19(24-17)21(29)23-12(11-25)8-18(26)27/h1-7,9,12,25,28H,8,11H2,(H,23,29)(H,26,27)/t12-/m1/s1
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n/an/a 1.59E+5n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240978
PNG
(US9409892, 73)
Show SMILES C[C@](O)(CNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)C(O)=O |r|
Show InChI InChI=1S/C21H17N3O6/c1-21(29,20(27)28)11-23-19(26)17-18(25)14-8-7-13(9-15(14)16(10-22)24-17)30-12-5-3-2-4-6-12/h2-9,25,29H,11H2,1H3,(H,23,26)(H,27,28)/t21-/m0/s1
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n/an/a 740n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240980
PNG
(US9409892, 75)
Show SMILES O[C@H]([C@@H](Cc1ccccc1)NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)C(O)=O |r|
Show InChI InChI=1S/C27H21N3O6/c28-15-22-20-14-18(36-17-9-5-2-6-10-17)11-12-19(20)24(31)23(29-22)26(33)30-21(25(32)27(34)35)13-16-7-3-1-4-8-16/h1-12,14,21,25,31-32H,13H2,(H,30,33)(H,34,35)/t21-,25-/m1/s1
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n/an/a 1.17E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241002
PNG
(US9409892, 97)
Show SMILES OC(=O)CCNC(=O)c1nc(C#N)c2cc(Oc3ccc(F)cc3Cl)ccc2c1O
Show InChI InChI=1S/C20H13ClFN3O5/c21-14-7-10(22)1-4-16(14)30-11-2-3-12-13(8-11)15(9-23)25-18(19(12)28)20(29)24-6-5-17(26)27/h1-4,7-8,28H,5-6H2,(H,24,29)(H,26,27)
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n/an/a 1.30E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241019
PNG
(US9409892, 114)
Show SMILES OC(=O)CCCCNC(=O)c1ncc2cc(Sc3ccccc3)ccc2c1O
Show InChI InChI=1S/C21H20N2O4S/c24-18(25)8-4-5-11-22-21(27)19-20(26)17-10-9-16(12-14(17)13-23-19)28-15-6-2-1-3-7-15/h1-3,6-7,9-10,12-13,26H,4-5,8,11H2,(H,22,27)(H,24,25)
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n/an/a 1.35E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241037
PNG
(US9409892, 132)
Show SMILES OC(=O)CCNC(=O)c1ncc2cc(ccc2c1O)-c1ccc(F)cc1
Show InChI InChI=1S/C19H15FN2O4/c20-14-4-1-11(2-5-14)12-3-6-15-13(9-12)10-22-17(18(15)25)19(26)21-8-7-16(23)24/h1-6,9-10,25H,7-8H2,(H,21,26)(H,23,24)
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n/an/a 2.38E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241040
PNG
(US9409892, 135)
Show SMILES OC(=O)CCNC(=O)c1ncc2cc(ccc2c1O)S(=O)(=O)C1CCCCC1
Show InChI InChI=1S/C19H22N2O6S/c22-16(23)8-9-20-19(25)17-18(24)15-7-6-14(10-12(15)11-21-17)28(26,27)13-4-2-1-3-5-13/h6-7,10-11,13,24H,1-5,8-9H2,(H,20,25)(H,22,23)
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n/an/a 350n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240966
PNG
(US9409892, 61)
Show SMILES CC(C)[C@H](NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)C(C)(C)C(O)=O |r|
Show InChI InChI=1S/C25H25N3O5/c1-14(2)22(25(3,4)24(31)32)28-23(30)20-21(29)17-11-10-16(12-18(17)19(13-26)27-20)33-15-8-6-5-7-9-15/h5-12,14,22,29H,1-4H3,(H,28,30)(H,31,32)/t22-/m0/s1
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n/an/a>2.00E+5n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240981
PNG
(US9409892, 76)
Show SMILES OC(CNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C20H15N3O6/c21-9-15-14-8-12(29-11-4-2-1-3-5-11)6-7-13(14)18(25)17(23-15)19(26)22-10-16(24)20(27)28/h1-8,16,24-25H,10H2,(H,22,26)(H,27,28)
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n/an/a 2.86E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240983
PNG
(US9409892, 78)
Show SMILES C[C@@H](CC(O)=O)NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O |r|
Show InChI InChI=1S/C21H17N3O5/c1-12(9-18(25)26)23-21(28)19-20(27)15-8-7-14(10-16(15)17(11-22)24-19)29-13-5-3-2-4-6-13/h2-8,10,12,27H,9H2,1H3,(H,23,28)(H,25,26)/t12-/m0/s1
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n/an/a 9.68E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240997
PNG
(US9409892, 92)
Show SMILES C[C@H](CNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)C(O)=O |r|
Show InChI InChI=1S/C21H17N3O5/c1-12(21(27)28)11-23-20(26)18-19(25)15-8-7-14(9-16(15)17(10-22)24-18)29-13-5-3-2-4-6-13/h2-9,12,25H,11H2,1H3,(H,23,26)(H,27,28)/t12-/m1/s1
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n/an/a 3.88E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241002
PNG
(US9409892, 97)
Show SMILES OC(=O)CCNC(=O)c1nc(C#N)c2cc(Oc3ccc(F)cc3Cl)ccc2c1O
Show InChI InChI=1S/C20H13ClFN3O5/c21-14-7-10(22)1-4-16(14)30-11-2-3-12-13(8-11)15(9-23)25-18(19(12)28)20(29)24-6-5-17(26)27/h1-4,7-8,28H,5-6H2,(H,24,29)(H,26,27)
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n/an/a 7.43E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241003
PNG
(US9409892, 98)
Show SMILES OC(=O)CCCCNC(=O)c1nc(C#N)c2cc(Oc3ccc(F)cc3Cl)ccc2c1O
Show InChI InChI=1S/C22H17ClFN3O5/c23-16-9-12(24)4-7-18(16)32-13-5-6-14-15(10-13)17(11-25)27-20(21(14)30)22(31)26-8-2-1-3-19(28)29/h4-7,9-10,30H,1-3,8H2,(H,26,31)(H,28,29)
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n/an/a 3.73E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241014
PNG
(US9409892, 109)
Show SMILES Cc1cccc(C)c1Oc1ccc2c(nc(C(=O)NCCC(O)=O)c(O)c2c1)C#N
Show InChI InChI=1S/C22H19N3O5/c1-12-4-3-5-13(2)21(12)30-14-6-7-15-16(10-14)20(28)19(25-17(15)11-23)22(29)24-9-8-18(26)27/h3-7,10,28H,8-9H2,1-2H3,(H,24,29)(H,26,27)
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n/an/a 3.04E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241018
PNG
(US9409892, 113)
Show SMILES OC(=O)CCCNC(=O)c1ncc2ccc(Oc3ccccc3)cc2c1O
Show InChI InChI=1S/C20H18N2O5/c23-17(24)7-4-10-21-20(26)18-19(25)16-11-15(9-8-13(16)12-22-18)27-14-5-2-1-3-6-14/h1-3,5-6,8-9,11-12,25H,4,7,10H2,(H,21,26)(H,23,24)
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n/an/a 2.00E+5n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241020
PNG
(US9409892, 115)
Show SMILES OC(=O)CCCNC(=O)c1ncc2cc(Sc3ccccc3)ccc2c1O
Show InChI InChI=1S/C20H18N2O4S/c23-17(24)7-4-10-21-20(26)18-19(25)16-9-8-15(11-13(16)12-22-18)27-14-5-2-1-3-6-14/h1-3,5-6,8-9,11-12,25H,4,7,10H2,(H,21,26)(H,23,24)
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n/an/a 1.48E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241035
PNG
(US9409892, 130)
Show SMILES OC(=O)CCNC(=O)c1ncc2cc(NC(=O)NC3CCCCC3)ccc2c1O
Show InChI InChI=1S/C20H24N4O5/c25-16(26)8-9-21-19(28)17-18(27)15-7-6-14(10-12(15)11-22-17)24-20(29)23-13-4-2-1-3-5-13/h6-7,10-11,13,27H,1-5,8-9H2,(H,21,28)(H,25,26)(H2,23,24,29)
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n/an/a 3.96E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241036
PNG
(US9409892, 131)
Show SMILES OC(=O)CCCNC(=O)c1ncc2cc(NC(=O)NC3CCCCC3)ccc2c1O
Show InChI InChI=1S/C21H26N4O5/c26-17(27)7-4-10-22-20(29)18-19(28)16-9-8-15(11-13(16)12-23-18)25-21(30)24-14-5-2-1-3-6-14/h8-9,11-12,14,28H,1-7,10H2,(H,22,29)(H,26,27)(H2,24,25,30)
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n/an/a 7.76E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241045
PNG
(US9409892, 140)
Show SMILES CC(C)(CNC(=O)c1nc(C#N)c2cc(NC(=O)Nc3ccccc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C23H21N5O5/c1-23(2,21(31)32)12-25-20(30)18-19(29)15-9-8-14(10-16(15)17(11-24)28-18)27-22(33)26-13-6-4-3-5-7-13/h3-10,29H,12H2,1-2H3,(H,25,30)(H,31,32)(H2,26,27,33)
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n/an/a 3.35E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241047
PNG
(US9409892, 142)
Show SMILES OC(=O)CCCNC(=O)c1ncc2cc(NC(=O)Nc3ccc(F)cc3)ccc2c1O
Show InChI InChI=1S/C21H19FN4O5/c22-13-3-5-14(6-4-13)25-21(31)26-15-7-8-16-12(10-15)11-24-18(19(16)29)20(30)23-9-1-2-17(27)28/h3-8,10-11,29H,1-2,9H2,(H,23,30)(H,27,28)(H2,25,26,31)
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n/an/a 5.64E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241056
PNG
(US9409892, 151)
Show SMILES Cn1nc(cc1-c1nc(C(=O)NCC(C)(C)C(O)=O)c(O)c2ccc(Oc3ccccc3)cc12)C(F)(F)F
Show InChI InChI=1S/C26H23F3N4O5/c1-25(2,24(36)37)13-30-23(35)21-22(34)16-10-9-15(38-14-7-5-4-6-8-14)11-17(16)20(31-21)18-12-19(26(27,28)29)32-33(18)3/h4-12,34H,13H2,1-3H3,(H,30,35)(H,36,37)
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n/an/a 1.11E+5n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241060
PNG
(US9409892, 155)
Show SMILES Cc1ccccc1Oc1ccc2c(nc(C(=O)NCC(C)(C)C(O)=O)c(O)c2c1)C#N
Show InChI InChI=1S/C23H21N3O5/c1-13-6-4-5-7-18(13)31-14-8-9-15-16(10-14)20(27)19(26-17(15)11-24)21(28)25-12-23(2,3)22(29)30/h4-10,27H,12H2,1-3H3,(H,25,28)(H,29,30)
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n/an/a 4.21E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241072
PNG
(US9409892, 167)
Show SMILES OC(=O)C(CNC(=O)c1ncc2cc(Oc3ccccc3)ccc2c1O)C1CC1
Show InChI InChI=1S/C22H20N2O5/c25-20-17-9-8-16(29-15-4-2-1-3-5-15)10-14(17)11-23-19(20)21(26)24-12-18(22(27)28)13-6-7-13/h1-5,8-11,13,18,25H,6-7,12H2,(H,24,26)(H,27,28)
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n/an/a 1.00E+5n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241077
PNG
(US9409892, 172)
Show SMILES OC(=O)C[C@H](NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)c1ccc(cc1)C#N |r|
Show InChI InChI=1S/C27H18N4O5/c28-14-16-6-8-17(9-7-16)22(13-24(32)33)31-27(35)25-26(34)20-11-10-19(12-21(20)23(15-29)30-25)36-18-4-2-1-3-5-18/h1-12,22,34H,13H2,(H,31,35)(H,32,33)/t22-/m0/s1
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n/an/a 2.76E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM241088
PNG
(US9409892, 183)
Show SMILES CC(C)CC(CNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)CC(O)=O
Show InChI InChI=1S/C25H25N3O5/c1-15(2)10-16(11-22(29)30)14-27-25(32)23-24(31)19-9-8-18(12-20(19)21(13-26)28-23)33-17-6-4-3-5-7-17/h3-9,12,15-16,31H,10-11,14H2,1-2H3,(H,27,32)(H,29,30)
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n/an/a 1.26E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240928
PNG
(US9409892, 23)
Show SMILES CC(C)(CNC(=O)c1ncc2cc(Oc3ccc(Cl)c(F)c3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C21H18ClFN2O5/c1-21(2,20(28)29)10-25-19(27)17-18(26)14-5-3-12(7-11(14)9-24-17)30-13-4-6-15(22)16(23)8-13/h3-9,26H,10H2,1-2H3,(H,25,27)(H,28,29)
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n/an/a 2.77E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240939
PNG
(US9409892, 34)
Show SMILES OC(=O)CC(CNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)c1ccc(Cl)cc1 |w:4.31|
Show InChI InChI=1S/C27H20ClN3O5/c28-18-8-6-16(7-9-18)17(12-24(32)33)15-30-27(35)25-26(34)21-11-10-20(13-22(21)23(14-29)31-25)36-19-4-2-1-3-5-19/h1-11,13,17,34H,12,15H2,(H,30,35)(H,32,33)
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n/an/a 2.55E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240952
PNG
(US9409892, 47)
Show SMILES OC(=O)C[C@H](NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)c1ccccc1 |r|
Show InChI InChI=1S/C26H19N3O5/c27-15-22-20-13-18(34-17-9-5-2-6-10-17)11-12-19(20)25(32)24(28-22)26(33)29-21(14-23(30)31)16-7-3-1-4-8-16/h1-13,21,32H,14H2,(H,29,33)(H,30,31)/t21-/m0/s1
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n/an/a 1.28E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM240958
PNG
(US9409892, 53)
Show SMILES COC(=O)NC(CCNC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C23H20N4O7/c1-33-23(32)27-17(22(30)31)9-10-25-21(29)19-20(28)15-8-7-14(11-16(15)18(12-24)26-19)34-13-5-3-2-4-6-13/h2-8,11,17,28H,9-10H2,1H3,(H,25,29)(H,27,32)(H,30,31)
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n/an/a 240n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241048
PNG
(US9409892, 143)
Show SMILES CC(C)(CNC(=O)c1nc(-c2ccccc2)c2cc(Oc3ccccc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C27H24N2O5/c1-27(2,26(32)33)16-28-25(31)23-24(30)20-14-13-19(34-18-11-7-4-8-12-18)15-21(20)22(29-23)17-9-5-3-6-10-17/h3-15,30H,16H2,1-2H3,(H,28,31)(H,32,33)
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n/an/a 1.11E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241053
PNG
(US9409892, 148)
Show SMILES OC(=O)CCCNC(=O)c1ncc2cc(ccc2c1O)-c1ccc(F)cc1
Show InChI InChI=1S/C20H17FN2O4/c21-15-6-3-12(4-7-15)13-5-8-16-14(10-13)11-23-18(19(16)26)20(27)22-9-1-2-17(24)25/h3-8,10-11,26H,1-2,9H2,(H,22,27)(H,24,25)
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n/an/a 2.88E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241055
PNG
(US9409892, 150)
Show SMILES CC(C)(CNC(=O)c1ncc2cc(ccc2c1O)-c1ccc(F)cc1)C(O)=O
Show InChI InChI=1S/C21H19FN2O4/c1-21(2,20(27)28)11-24-19(26)17-18(25)16-8-5-13(9-14(16)10-23-17)12-3-6-15(22)7-4-12/h3-10,25H,11H2,1-2H3,(H,24,26)(H,27,28)
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n/an/a 2.29E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241069
PNG
(US9409892, 164)
Show SMILES CC(C)(CNC(=O)c1nc(C#N)c2cc(Cc3ccccc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C23H21N3O4/c1-23(2,22(29)30)13-25-21(28)19-20(27)16-9-8-15(10-14-6-4-3-5-7-14)11-17(16)18(12-24)26-19/h3-9,11,27H,10,13H2,1-2H3,(H,25,28)(H,29,30)
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n/an/a 1.35E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Prolyl hydroxylase EGLN2


(Homo sapiens (Human))		BDBM241070
PNG
(US9409892, 165)
Show SMILES OC(=O)CC(NC(=O)c1nc(C#N)c2cc(Oc3ccccc3)ccc2c1O)c1cccc(Cl)c1
Show InChI InChI=1S/C26H18ClN3O5/c27-16-6-4-5-15(11-16)21(13-23(31)32)30-26(34)24-25(33)19-10-9-18(12-20(19)22(14-28)29-24)35-17-7-2-1-3-8-17/h1-12,21,33H,13H2,(H,30,34)(H,31,32)
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n/an/a 1.51E+3n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240907
PNG
(US9409892, 2)
Show SMILES CC(C)(CNC(=O)c1ncc2cc(Oc3ccccc3)ccc2c1O)C(O)=O
Show InChI InChI=1S/C21H20N2O5/c1-21(2,20(26)27)12-23-19(25)17-18(24)16-9-8-15(10-13(16)11-22-17)28-14-6-4-3-5-7-14/h3-11,24H,12H2,1-2H3,(H,23,25)(H,26,27)
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n/an/a 4.67E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
Egl nine homolog 1


(Homo sapiens (Human))		BDBM240921
PNG
(US9409892, 16)
Show SMILES OC(=O)C1(CNC(=O)c2nc(C#N)c3cc(Oc4ccccc4)ccc3c2O)CCOCC1
Show InChI InChI=1S/C24H21N3O6/c25-13-19-18-12-16(33-15-4-2-1-3-5-15)6-7-17(18)21(28)20(27-19)22(29)26-14-24(23(30)31)8-10-32-11-9-24/h1-7,12,28H,8-11,14H2,(H,26,29)(H,30,31)
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n/an/a 2.43E+4n/an/an/an/a7.4n/a



FibroGen, Inc.

US Patent


Assay Description
Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources...

US Patent US9409892 (2016)


BindingDB Entry DOI: 10.7270/Q2MG7NFC
More data for this
Ligand-Target Pair
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* indicates data uncertainty>20%