Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106677 (US8586580, 25) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | <500 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106673 (US8586580, 1) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | <500 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106676 (US8586580, 13) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <500 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106679 (US8586580, 27) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | <500 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106680 (US8586580, 30) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <500 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106675 (US8586580, 12) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106674 (US8586580, 11) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Focal adhesion kinase 1 (Homo sapiens (Human)) | BDBM106678 (US8586580, 26) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Korea Institute of Science and Technology US Patent | Assay Description FAK kinase assay using ulight-LANCE assay purchased from PerkinElmer (catalog # TRF0100-D). | US Patent US8586580 (2013) BindingDB Entry DOI: 10.7270/Q2BP01FV | |||||||||||
More data for this Ligand-Target Pair |