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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223491 (US10407441, Compound JQ6 | US10925881, Name (S)-JQ...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet  | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.240 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223492 (US10407441, Compound JQ8 | US10925881, Name (S)-JQ...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.427 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223493 (US10407441, Compound JQ13 | US10925881, Name (S)-J...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.584 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223492 (US10407441, Compound JQ8 | US10925881, Name (S)-JQ...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.19 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223493 (US10407441, Compound JQ13 | US10925881, Name (S)-J...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.49 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223491 (US10407441, Compound JQ6 | US10925881, Name (S)-JQ...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.48 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223495 (US10407441, Compound JQ35 | US9320741, JQ35) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.13 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50365262 ((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50365262 ((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223495 (US10407441, Compound JQ35 | US9320741, JQ35) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 24.3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223494 (US10407441, Compound JQ33 | US9320741, JQ33) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 29.5 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM223494 (US10407441, Compound JQ33 | US9320741, JQ33) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 85 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM205429 ( (R)-JQ1 (3) | US10407441, Compound (R)-JQ1 | US10...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 8.35E+6 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM205429 ( (R)-JQ1 (3) | US10407441, Compound (R)-JQ1 | US10...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 5.21E+7 | n/a | n/a | n/a | n/a | 7.4 | 25 |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer... | US Patent US9320741 (2016) BindingDB Entry DOI: 10.7270/Q2KP811P | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
