Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (719/719 = 100%)† (Homo sapiens (Human)) | BDBM50118239 (CHEMBL130266 | UDP | Uridine diphosphate | uridine...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of British Columbia Curated by ChEMBL | Assay Description Inhibition of human OGT | Bioorg Med Chem Lett 21: 1199-201 (2011) Article DOI: 10.1016/j.bmcl.2010.12.090 BindingDB Entry DOI: 10.7270/Q2028RT6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |