Found 20 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Glutamate receptor 3
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 570 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85744
(ATPA-S)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15)/t6-/m1/s1 | PDB
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| 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar
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| PC cid
PC sid
UniChem
Similars
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
UniProtKB/SwissProt
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UniChem
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85741
(ATPA | CAS_140158-50-5 | NSC_2253)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15) | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85744
(ATPA-S)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15)/t6-/m1/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM50002370
((R,S)-alpha-amino-3-hydroxy-5-methyl-4-isooxazole-...)Show InChI InChI=1S/C7H10N2O4/c1-3-4(6(10)9-13-3)2-5(8)7(11)12/h5H,2,8H2,1H3,(H,9,10)(H,11,12) | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85744
(ATPA-S)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15)/t6-/m1/s1 | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
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UniChem
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
UniProtKB/SwissProt
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| PC cid
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UniChem
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85741
(ATPA | CAS_140158-50-5 | NSC_2253)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15) | PDB
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85742
(ATPA-R)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15)/t6-/m0/s1 | PDB
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85743
(CAS_5289517 | NSC_5289517 | Thio-ATPA | Thio-ATPA-...)Show InChI InChI=1S/C10H16N2O3S/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H2,12,13,14,15) | PDB
UniProtKB/SwissProt
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85741
(ATPA | CAS_140158-50-5 | NSC_2253)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15) | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM85742
(ATPA-R)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15)/t6-/m0/s1 | PDB
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM85742
(ATPA-R)Show InChI InChI=1S/C10H16N2O4/c1-10(2,3)7-5(8(13)12-16-7)4-6(11)9(14)15/h6H,4,11H2,1-3H3,(H,12,13)(H,14,15)/t6-/m0/s1 | PDB
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PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM50002370
((R,S)-alpha-amino-3-hydroxy-5-methyl-4-isooxazole-...)Show InChI InChI=1S/C7H10N2O4/c1-3-4(6(10)9-13-3)2-5(8)7(11)12/h5H,2,8H2,1H3,(H,9,10)(H,11,12) | PDB
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy
Curated by PDSP Ki Database
| |
Eur J Pharmacol 411: 245-53 (2001)
Article DOI: 10.1016/s0014-2999(00)00916-x
BindingDB Entry DOI: 10.7270/Q2G73C8N |
More data for this
Ligand-Target Pair | |
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