Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gamma-aminobutyric acid receptor subunit alpha-1 (Mus musculus) | BDBM50001561 (5-(6-Imino-3-thiophen-3-yl-6H-pyridazin-1-ylmethyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 88 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations. | J Med Chem 35: 4092-7 (1992) BindingDB Entry DOI: 10.7270/Q25X29J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1 (Mus musculus) | BDBM50001562 (5-(6-Imino-3-phenyl-6H-pyridazin-1-ylmethyl)-isoxa...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations. | J Med Chem 35: 4092-7 (1992) BindingDB Entry DOI: 10.7270/Q25X29J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1 (Mus musculus) | BDBM50001556 (4-(6-Imino-5-methyl-3-phenyl-6H-pyridazin-1-yl)-bu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations. | J Med Chem 35: 4092-7 (1992) BindingDB Entry DOI: 10.7270/Q25X29J4 | |||||||||||
More data for this Ligand-Target Pair |