Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholecystokinin receptor type A (RAT) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060319 (CHEMBL113718 | [(S)-1-((4aS,5R)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.59 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S348A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (M195L) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S348A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (M195L) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1R | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S342A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1R | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R197M) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11.8 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R197M) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R197M) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (F107A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (T117A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26.8 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (F107A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 27.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S342A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (T117A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 31.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (F107A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 33.2 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S342A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35.2 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1R | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35.2 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (M195L) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 36.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S348A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 71.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (T117A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 129 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 183 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329F) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 227 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I352A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 514 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329F) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 582 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R336M) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 801 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329F) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 831 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I352A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R336M) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.29E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I352A) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.86E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R336M) | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50060322 (CHEMBL332261 | [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 2 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50060322 (CHEMBL332261 | [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50170765 (CHEMBL363916 | [(S)-1-((4aS,5R)-2-Benzyl-1-mercapt...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 2 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50170766 (CHEMBL189634 | [(S)-1-((4aS,5R)-1,3-Dioxo-2-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 2 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50170764 (CHEMBL366344 | [(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 2 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060319 (CHEMBL113718 | [(S)-1-((4aS,5R)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 2 receptor | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50060322 (CHEMBL332261 | [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.09E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1R | J Med Chem 48: 4842-50 (2005) Article DOI: 10.1021/jm0501127 BindingDB Entry DOI: 10.7270/Q2WQ03BN | |||||||||||
More data for this Ligand-Target Pair |