Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM92983 (MPP analogue, 19) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California, San Francisco | Assay Description Inhibition assay using MAO-A and MAO-B. | Biochemistry 31: 5611-5 (1992) Article DOI: 10.1021/bi00139a026 BindingDB Entry DOI: 10.7270/Q2RF5SNV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM92982 (MPP analogue, 18) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California, San Francisco | Assay Description Inhibition assay using MAO-A and MAO-B. | Biochemistry 31: 5611-5 (1992) Article DOI: 10.1021/bi00139a026 BindingDB Entry DOI: 10.7270/Q2RF5SNV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM92981 (MPP analogue, 17) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California, San Francisco | Assay Description Inhibition assay using MAO-A and MAO-B. | Biochemistry 31: 5611-5 (1992) Article DOI: 10.1021/bi00139a026 BindingDB Entry DOI: 10.7270/Q2RF5SNV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] B (Homo sapiens (Human)) | BDBM92981 (MPP analogue, 17) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California, San Francisco | Assay Description Inhibition assay using MAO-A and MAO-B. | Biochemistry 31: 5611-5 (1992) Article DOI: 10.1021/bi00139a026 BindingDB Entry DOI: 10.7270/Q2RF5SNV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] B (Homo sapiens (Human)) | BDBM92983 (MPP analogue, 19) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California, San Francisco | Assay Description Inhibition assay using MAO-A and MAO-B. | Biochemistry 31: 5611-5 (1992) Article DOI: 10.1021/bi00139a026 BindingDB Entry DOI: 10.7270/Q2RF5SNV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] B (Homo sapiens (Human)) | BDBM92982 (MPP analogue, 18) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California, San Francisco | Assay Description Inhibition assay using MAO-A and MAO-B. | Biochemistry 31: 5611-5 (1992) Article DOI: 10.1021/bi00139a026 BindingDB Entry DOI: 10.7270/Q2RF5SNV | |||||||||||
More data for this Ligand-Target Pair |