Affinity Data by PubMed id=17918820

PubMed code 17918820

Found 6 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Estrogen receptor (Homo sapiens (Human))	BDBM50224172 (CHEMBL235496 \| methyl 4-(4-(2-fluorobenzyloxy)phen...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	53	n/a	n/a	n/a	n/a	n/a	n/a
Trinity College Curated by ChEMBL					Assay Description Displacement of fluoromone from human recombinant ERalpha by fluorescence polarization assay				J Med Chem 50: 5301-10 (2007) Article DOI: 10.1021/jm0700262 BindingDB Entry DOI: 10.7270/Q2F47NW6
Trinity College Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50224174 (2-amino-7-hydroxy-4-[4-(4-methyl-benzyloxy)-phenyl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	56	n/a	n/a	n/a	n/a	n/a	n/a
Trinity College Curated by ChEMBL					Assay Description Displacement of fluoromone from human recombinant ERalpha by fluorescence polarization assay				J Med Chem 50: 5301-10 (2007) Article DOI: 10.1021/jm0700262 BindingDB Entry DOI: 10.7270/Q2F47NW6
Trinity College Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor beta (Homo sapiens (Human))	BDBM50224172 (CHEMBL235496 \| methyl 4-(4-(2-fluorobenzyloxy)phen...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	780	n/a	n/a	n/a	n/a	n/a	n/a
Trinity College Curated by ChEMBL					Assay Description Displacement of fluoromone from human recombinant ERbeta by fluorescence polarization assay				J Med Chem 50: 5301-10 (2007) Article DOI: 10.1021/jm0700262 BindingDB Entry DOI: 10.7270/Q2F47NW6
Trinity College Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor beta (Homo sapiens (Human))	BDBM50224174 (2-amino-7-hydroxy-4-[4-(4-methyl-benzyloxy)-phenyl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	915	n/a	n/a	n/a	n/a	n/a	n/a
Trinity College Curated by ChEMBL					Assay Description Displacement of fluoromone from human recombinant ERbeta by fluorescence polarization assay				J Med Chem 50: 5301-10 (2007) Article DOI: 10.1021/jm0700262 BindingDB Entry DOI: 10.7270/Q2F47NW6
Trinity College Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50224173 (3-benzyl-2-(4-hydroxy-3-methoxyphenyl)-2,3-dihydro...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
Trinity College Curated by ChEMBL					Assay Description Displacement of fluoromone from human recombinant ERalpha by fluorescence polarization assay				J Med Chem 50: 5301-10 (2007) Article DOI: 10.1021/jm0700262 BindingDB Entry DOI: 10.7270/Q2F47NW6
Trinity College Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor beta (Homo sapiens (Human))	BDBM50224173 (3-benzyl-2-(4-hydroxy-3-methoxyphenyl)-2,3-dihydro...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
Trinity College Curated by ChEMBL					Assay Description Displacement of fluoromone from human recombinant ERbeta by fluorescence polarization assay				J Med Chem 50: 5301-10 (2007) Article DOI: 10.1021/jm0700262 BindingDB Entry DOI: 10.7270/Q2F47NW6
Trinity College Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%