Affinity Data by PubMed id=17931863

PubMed code 17931863

Found 2 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Hydroxycarboxylic acid receptor 2 (Homo sapiens (Human))	BDBM50224535 (6-(pentan-3-ylamino)nicotinic acid \| CHEMBL396879) Show SMILES CCC(CC)Nc1ccc(cn1)C(O)=O Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a
Arena Pharmaceuticals Curated by ChEMBL					Assay Description Agonist activity at human GPR109a receptor transfected in CHOK1 cells assessed as reversal of forskolin induced cAMP elevating effect by whole cell a...				Bioorg Med Chem Lett 17: 6619-22 (2007) Article DOI: 10.1016/j.bmcl.2007.09.058 BindingDB Entry DOI: 10.7270/Q20V8CHJ
Arena Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair
Hydroxycarboxylic acid receptor 2 (Homo sapiens (Human))	BDBM50224534 (6-(isobutylamino)nicotinic acid \| CHEMBL237737) Show SMILES CC(C)CNc1ccc(cn1)C(O)=O Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	3.50E+4	n/a	n/a	n/a	n/a
Arena Pharmaceuticals Curated by ChEMBL					Assay Description Agonist activity at human GPR109a receptor transfected in CHOK1 cells assessed as reversal of forskolin induced cAMP elevating effect by whole cell a...				Bioorg Med Chem Lett 17: 6619-22 (2007) Article DOI: 10.1016/j.bmcl.2007.09.058 BindingDB Entry DOI: 10.7270/Q20V8CHJ
Arena Pharmaceuticals Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%