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PubMed code 18665581

Compile data set for download or QSAR
Found 23 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273030
PNG
((E)-2-(5-Fluoro-1-(naphthalen-1-ylmethylene)-1H-in...)
Show SMILES OC(=O)CC1=C\C(=C/c2cccc3ccccc23)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C22H15FO2/c23-18-8-9-20-16(11-17(12-22(24)25)21(20)13-18)10-15-6-3-5-14-4-1-2-7-19(14)15/h1-11,13H,12H2,(H,24,25)/b16-10+
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n/an/an/an/a 100n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272984
PNG
((E)-2-(5-Fluoro-1-(4-(trifluoromethyl)benzylidene)...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(cc2)C(F)(F)F)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C19H12F4O2/c20-15-5-6-16-12(8-13(9-18(24)25)17(16)10-15)7-11-1-3-14(4-2-11)19(21,22)23/h1-8,10H,9H2,(H,24,25)/b12-7+
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n/an/an/an/a 2.50E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272985
PNG
((E)-2-(1-(4-Ethynylbenzylidene)-5-fluoro-1H-inden-...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(cc2)C#C)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C20H13FO2/c1-2-13-3-5-14(6-4-13)9-15-10-16(11-20(22)23)19-12-17(21)7-8-18(15)19/h1,3-10,12H,11H2,(H,22,23)/b15-9+
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n/an/an/an/a 1.10E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272902
PNG
((E)-4-((3-(Carboxymethyl)-5-fluoro-1H-inden-1-ylid...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(cc2)C(O)=O)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C19H13FO4/c20-15-5-6-16-13(8-14(9-18(21)22)17(16)10-15)7-11-1-3-12(4-2-11)19(23)24/h1-8,10H,9H2,(H,21,22)(H,23,24)/b13-7+
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n/an/an/an/a>1.00E+4n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273031
PNG
((E)-2-(5-Fluoro-1-((4-fluoronaphthalen-1-yl)methyl...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(F)c3ccccc23)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C22H14F2O2/c23-16-6-7-18-14(10-15(11-22(25)26)20(18)12-16)9-13-5-8-21(24)19-4-2-1-3-17(13)19/h1-10,12H,11H2,(H,25,26)/b14-9+
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n/an/an/an/a 100n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272988
PNG
((E)-2-(1-(4-tert-Butoxybenzylidene)-5-fluoro-1H-in...)
Show SMILES CC(C)(C)Oc1ccc(\C=C2/C=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:11|
Show InChI InChI=1S/C22H21FO3/c1-22(2,3)26-18-7-4-14(5-8-18)10-15-11-16(12-21(24)25)20-13-17(23)6-9-19(15)20/h4-11,13H,12H2,1-3H3,(H,24,25)/b15-10+
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n/an/an/an/a 1.90E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272986
PNG
((E)-2-(1-(4-(Azidomethyl)benzylidene)-5-fluoro-1H-...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(CN=[N+]=[N-])cc2)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C19H14FN3O2/c20-16-5-6-17-14(8-15(9-19(24)25)18(17)10-16)7-12-1-3-13(4-2-12)11-22-23-21/h1-8,10H,9,11H2,(H,24,25)/b14-7+
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n/an/an/an/a 900n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272906
PNG
((E)-2-(5-Fluoro-1-(4-methylbenzylidene)-1H-inden-3...)
Show SMILES Cc1ccc(\C=C2/C=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:7|
Show InChI InChI=1S/C19H15FO2/c1-12-2-4-13(5-3-12)8-14-9-15(10-19(21)22)18-11-16(20)6-7-17(14)18/h2-9,11H,10H2,1H3,(H,21,22)/b14-8+
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n/an/an/an/a 2.40E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272905
PNG
((E)-2-(1-Benzylidene-5-fluoro-1H-inden-3-yl)ethano...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccccc2)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C18H13FO2/c19-15-6-7-16-13(8-12-4-2-1-3-5-12)9-14(10-18(20)21)17(16)11-15/h1-9,11H,10H2,(H,20,21)/b13-8+
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n/an/an/an/a 1.70E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273067
PNG
((E)-2-(1-((2,4-Difluorobiphenyl-4-yl)methylene)-5-...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(cc2)-c2ccc(F)cc2F)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C24H15F3O2/c25-18-5-7-20-16(10-17(11-24(28)29)22(20)12-18)9-14-1-3-15(4-2-14)21-8-6-19(26)13-23(21)27/h1-10,12-13H,11H2,(H,28,29)/b16-9+
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n/an/an/an/a 100n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273065
PNG
((E)-2-(1-(Biphenyl-4-ylmethylene)-5-fluoro-1H-inde...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(cc2)-c2ccccc2)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C24H17FO2/c25-21-10-11-22-19(13-20(14-24(26)27)23(22)15-21)12-16-6-8-18(9-7-16)17-4-2-1-3-5-17/h1-13,15H,14H2,(H,26,27)/b19-12+
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n/an/an/an/a 100n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273064
PNG
((E)-2-(5-Fluoro-1-(quinolin-8-ylmethylene)-1H-inde...)
Show SMILES OC(=O)CC1=C\C(=C/c2cccc3cccnc23)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C21H14FNO2/c22-17-6-7-18-15(10-16(11-20(24)25)19(18)12-17)9-14-4-1-3-13-5-2-8-23-21(13)14/h1-10,12H,11H2,(H,24,25)/b15-9+
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n/an/an/an/a 1.50E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272861
PNG
((E)-2-(5-Fluoro-1-(4-(methylsulfinyl)benzylidene)-...)
Show SMILES CS(=O)c1ccc(\C=C2/C=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:9|
Show InChI InChI=1S/C19H15FO3S/c1-24(23)16-5-2-12(3-6-16)8-13-9-14(10-19(21)22)18-11-15(20)4-7-17(13)18/h2-9,11H,10H2,1H3,(H,21,22)/b13-8+
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n/an/an/an/a>1.00E+4n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272862
PNG
((E)-2'-des-methyl sulindac sulfide | 2-desmethylsu...)
Show SMILES CSc1ccc(\C=C2/C=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:8|
Show InChI InChI=1S/C19H15FO2S/c1-23-16-5-2-12(3-6-16)8-13-9-14(10-19(21)22)18-11-15(20)4-7-17(13)18/h2-9,11H,10H2,1H3,(H,21,22)/b13-8+
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n/an/an/an/a 700n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50110164
PNG
((Z)-2-(3-(4-(methylthio)benzylidene)-6-fluoro-2-me...)
Show SMILES CSc1ccc(\C=C2\C(C)=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:9|
Show InChI InChI=1S/C20H17FO2S/c1-12-17(9-13-3-6-15(24-2)7-4-13)16-8-5-14(21)10-19(16)18(12)11-20(22)23/h3-10H,11H2,1-2H3,(H,22,23)/b17-9-
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n/an/an/an/a 800n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair		3D
3D Structure (crystal)
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273028
PNG
((E)-2-(5-Fluoro-1-(naphthalen-2-ylmethylene)-1H-in...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc3ccccc3c2)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C22H15FO2/c23-19-7-8-20-17(11-18(12-22(24)25)21(20)13-19)10-14-5-6-15-3-1-2-4-16(15)9-14/h1-11,13H,12H2,(H,24,25)/b17-10+
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n/an/an/an/a 1.20E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273027
PNG
((E)-2-(5-Fluoro-1-(4-(trifluoromethylthio)benzylid...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(SC(F)(F)F)cc2)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C19H12F4O2S/c20-14-3-6-16-12(8-13(9-18(24)25)17(16)10-14)7-11-1-4-15(5-2-11)26-19(21,22)23/h1-8,10H,9H2,(H,24,25)/b12-7+
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n/an/an/an/a 200n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272987
PNG
((E)-2-(5-Fluoro-1-(4-methoxybenzylidene)-1H-inden-...)
Show SMILES COc1ccc(\C=C2/C=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:8|
Show InChI InChI=1S/C19H15FO3/c1-23-16-5-2-12(3-6-16)8-13-9-14(10-19(21)22)18-11-15(20)4-7-17(13)18/h2-9,11H,10H2,1H3,(H,21,22)/b13-8+
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PubMed
n/an/an/an/a 1.30E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272903
PNG
((E)-2-(1-(4-Bromobenzylidene)-5-fluoro-1H-inden-3-...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc(Br)cc2)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C18H12BrFO2/c19-14-3-1-11(2-4-14)7-12-8-13(9-18(21)22)17-10-15(20)5-6-16(12)17/h1-8,10H,9H2,(H,21,22)/b12-7+
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PubMed
n/an/an/an/a 1.10E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272904
PNG
(2-(5-Fluoro-1H-inden-3-yl)ethanoic acid | CHEMBL50...)
Show SMILES OC(=O)CC1=CCc2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C11H9FO2/c12-9-4-3-7-1-2-8(5-11(13)14)10(7)6-9/h2-4,6H,1,5H2,(H,13,14)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50272901
PNG
((E)-2-(5-Fluoro-1-(4-(methylsulfonyl)benzylidene)-...)
Show SMILES CS(=O)(=O)c1ccc(\C=C2/C=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:10|
Show InChI InChI=1S/C19H15FO4S/c1-25(23,24)16-5-2-12(3-6-16)8-13-9-14(10-19(21)22)18-11-15(20)4-7-17(13)18/h2-9,11H,10H2,1H3,(H,21,22)/b13-8+
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n/an/an/an/a>1.00E+4n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273066
PNG
((E)-2-(5-Fluoro-1-((4-(methylthio)biphenyl-4-yl)me...)
Show SMILES CSc1ccc(cc1)-c1ccc(\C=C2/C=C(CC(O)=O)c3cc(F)ccc23)cc1 |t:15|
Show InChI InChI=1S/C25H19FO2S/c1-29-22-9-6-18(7-10-22)17-4-2-16(3-5-17)12-19-13-20(14-25(27)28)24-15-21(26)8-11-23(19)24/h2-13,15H,14H2,1H3,(H,27,28)/b19-12+
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n/an/an/an/a 1.50E+3n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50273029
PNG
((E)-2-(5-Fluoro-1-(quinoxalin-6-ylmethylene)-1H-in...)
Show SMILES OC(=O)CC1=C\C(=C/c2ccc3nccnc3c2)c2ccc(F)cc12 |t:4|
Show InChI InChI=1S/C20H13FN2O2/c21-15-2-3-16-13(9-14(10-20(24)25)17(16)11-15)7-12-1-4-18-19(8-12)23-6-5-22-18/h1-9,11H,10H2,(H,24,25)/b13-7+
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n/an/an/an/a>1.00E+4n/an/an/an/a



Vanderbilt University Center for Structural Biology

Curated by ChEMBL


Assay Description
Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...

J Med Chem 51: 4911-9 (2008)


Article DOI: 10.1021/jm700969c
BindingDB Entry DOI: 10.7270/Q2H70FM4
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%