Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275728 (CHEMBL486749 | N-(4-chlorophenethyl)-2-isobutyl-N-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275896 (CHEMBL471017 | ethyl 2-(N-(1,4-dioxaspiro[4.5]deca...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275644 (CHEMBL520715 | cis-N-(4-chlorophenethyl)-N-(1-oxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275729 (CHEMBL486953 | N-(4-chlorophenethyl)-2-ethyl-N-(1,...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50266070 (4-(N-(4-chlorophenethyl)benzo[b]thiophene-3-carbox...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275779 (CHEMBL471210 | N-(2-(4-chlorophenyl)propyl)-N-(1,4...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275573 (CHEMBL487167 | trans-N-(4-chlorophenethyl)-N-4-hyd...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275605 (CHEMBL519540 | N-(4-chlorophenethyl)-N-(1,4-dioxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275683 (CHEMBL488388 | N-(4-chlorophenethyl)-N-(1,4-dioxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275897 (CHEMBL471018 | methyl 2-(N-(1,4-dioxaspiro[4.5]dec...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275834 (CHEMBL469527 | N-(2-(4-chlorophenyl)-2-methylpropy...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275777 (CHEMBL471009 | N-(4-chlorophenethyl)-N-(1,4-dioxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50266071 (CHEMBL518254 | N-(4-chlorophenethyl)-N-((1r,4r)-4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 125 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275727 (CHEMBL486748 | N-(4-chlorophenethyl)-2-(methoxymet...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 175 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275608 (CHEMBL485769 | N-(4-chlorophenethyl)-N-cyclohexylb...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 175 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275645 (CHEMBL487141 | trans-N-(4-chlorophenethyl)-N-(1-ox...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275570 (CHEMBL519730 | N-(4-chlorophenethyl)-N-(1-(2,4-dif...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275604 (CHEMBL485766 | cis-N-(4-chlorophenethyl)-N-(4-hydr...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275898 (CHEMBL470384 | methyl 2-(N-(1,4-dioxaspiro[4.5]dec...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275778 (CHEMBL513055 | N-(2-chlorophenethyl)-N-(1,4-dioxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275539 (CHEMBL519401 | N-(4-chlorophenethyl)-N-(1-(2-(2,4-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275572 (CHEMBL486971 | N-(4-chlorophenethyl)-N-(4-oxocyclo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275643 (CHEMBL519705 | N-benzyl-N-(4-chlorophenethyl)benzo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275833 (CHEMBL511613 | N-benzyl-N-(1,4-dioxaspiro[4.5]deca...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 395 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275776 (CHEMBL513247 | N-(4-chlorophenethyl)-N-(1,4-dioxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275835 (CHEMBL469528 | N-(2-(4-chlorophenoxy)ethyl)-N-(1,4...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 435 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275726 (CHEMBL520381 | N-(4-chlorophenethyl)-2-isopropoxy-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 835 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275538 (CHEMBL486959 | CP-289503 | N-(4-chlorophenethyl)-N...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275606 (CHEMBL485767 | N-(6-aminopyridin-3-yl)-N-(4-chloro...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275646 (CHEMBL487142 | N-(4-chlorophenethyl)-N-(1,4-dioxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275607 (CHEMBL488185 | N-(4-chlorophenethyl)-N-(tetrahydro...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275832 (CHEMBL512477 | N-(2-(pyridin-2-yl)ethyl)-N-(1,4-di...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275681 (CHEMBL519048 | N-(4-chlorophenethyl)-N-(1,4-dioxas...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275682 (CHEMBL528767 | N-(4-chlorophenethyl)-3-methoxy-N-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275684 (CHEMBL488389 | N-(4-chlorophenethyl)-2-(methylamin...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50275571 (CHEMBL486970 | N-(4-chlorophenethyl)-N-(piperidin-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cells | Bioorg Med Chem Lett 18: 5601-4 (2008) Article DOI: 10.1016/j.bmcl.2008.08.106 BindingDB Entry DOI: 10.7270/Q2TQ61CX | |||||||||||
More data for this Ligand-Target Pair |