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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Cathepsin K (Oryctolagus cuniculus (rabbit)) | BDBM19847 ((1R,2R)-N-(cyanomethyl)-5,5-difluoro-2-{2-[4-(meth...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.320 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Frosst Centre for Therapeutic Research Curated by ChEMBL | Assay Description Inhibition of rabbit cathepsin K | J Med Chem 51: 6410-20 (2008) Article DOI: 10.1021/jm800610j BindingDB Entry DOI: 10.7270/Q261105F | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cathepsin K (Oryctolagus cuniculus (rabbit)) | BDBM19909 ((1R,2R)-N-(cyanomethyl)-5,5-difluoro-2-{1-methyl-4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Frosst Centre for Therapeutic Research Curated by ChEMBL | Assay Description Inhibition of rabbit cathepsin K | J Med Chem 51: 6410-20 (2008) Article DOI: 10.1021/jm800610j BindingDB Entry DOI: 10.7270/Q261105F | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cathepsin K (Oryctolagus cuniculus (rabbit)) | BDBM50253069 ((1R,2R)-N-(1-cyanocyclopropyl)-5,5-difluoro-2-(1-m...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Frosst Centre for Therapeutic Research Curated by ChEMBL | Assay Description Inhibition of rabbit cathepsin K | J Med Chem 51: 6410-20 (2008) Article DOI: 10.1021/jm800610j BindingDB Entry DOI: 10.7270/Q261105F | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cathepsin K (Oryctolagus cuniculus (rabbit)) | BDBM50253098 ((1R,2R)-5,5-Dichloro-N-(1-cyanocyclopropyl)-2-[4-[...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Frosst Centre for Therapeutic Research Curated by ChEMBL | Assay Description Inhibition of rabbit cathepsin K | J Med Chem 51: 6410-20 (2008) Article DOI: 10.1021/jm800610j BindingDB Entry DOI: 10.7270/Q261105F | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cathepsin K (Oryctolagus cuniculus (rabbit)) | BDBM50253097 ((1R,2R)-N-(1-cyanocyclopropyl)-5,5-difluoro-2-(4-(...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Frosst Centre for Therapeutic Research Curated by ChEMBL | Assay Description Inhibition of rabbit cathepsin K | J Med Chem 51: 6410-20 (2008) Article DOI: 10.1021/jm800610j BindingDB Entry DOI: 10.7270/Q261105F | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cathepsin K (Oryctolagus cuniculus (rabbit)) | BDBM50253070 ((1R,2R)-N-(1-cyanocyclopropyl)-5,5-difluoro-2-(4-(...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Frosst Centre for Therapeutic Research Curated by ChEMBL | Assay Description Inhibition of rabbit cathepsin K | J Med Chem 51: 6410-20 (2008) Article DOI: 10.1021/jm800610j BindingDB Entry DOI: 10.7270/Q261105F | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
