Affinity Data by PubMed id=20207141

PubMed code 20207141

Found 2 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
C-C chemokine receptor type 5 (Homo sapiens (Human))	BDBM50314723 (CHEMBL1090041 \| endo-(S)-N-(4-fluorobenzyl)-4-(3-(...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	14.4	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Materia Medica Curated by ChEMBL					Assay Description Antagonist activity at CCR5 receptor expressed in CHO cells assessed as inhibition of RANTES-induced [32S]GTPgammaS binding				Bioorg Med Chem Lett 20: 2219-23 (2010) Article DOI: 10.1016/j.bmcl.2010.02.023 BindingDB Entry DOI: 10.7270/Q2C53M0B
Institute of Materia Medica Curated by ChEMBL					More data for this Ligand-Target Pair
C-C chemokine receptor type 5 (Homo sapiens (Human))	BDBM50314722 (CHEMBL1093331 \| endo-(S)-methyl 4-(3-(2-methyl-3H-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	112	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Materia Medica Curated by ChEMBL					Assay Description Antagonist activity at CCR5 receptor expressed in CHO cells assessed as inhibition of RANTES-induced [32S]GTPgammaS binding				Bioorg Med Chem Lett 20: 2219-23 (2010) Article DOI: 10.1016/j.bmcl.2010.02.023 BindingDB Entry DOI: 10.7270/Q2C53M0B
Institute of Materia Medica Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%