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PubMed code 20299214

Compile data set for download or QSAR
Found 20 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315313
PNG
((S)-2-(4-(4-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)S(=O)(=O)c2ccc(F)cc2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32FN3O6S/c1-22-28(33-30(41-22)24-5-3-2-4-6-24)15-20-40-26-11-7-23(8-12-26)21-29(31(36)37)34-16-18-35(19-17-34)42(38,39)27-13-9-25(32)10-14-27/h2-14,29H,15-21H2,1H3,(H,36,37)/t29-/m0/s1
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n/an/an/an/a 1.35E+3n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315312
PNG
((S)-2-(4-(2-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)S(=O)(=O)c2ccccc2F)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32FN3O6S/c1-22-27(33-30(41-22)24-7-3-2-4-8-24)15-20-40-25-13-11-23(12-14-25)21-28(31(36)37)34-16-18-35(19-17-34)42(38,39)29-10-6-5-9-26(29)32/h2-14,28H,15-21H2,1H3,(H,36,37)/t28-/m0/s1
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n/an/an/an/a 32n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315311
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)S(=O)(=O)c2ccccc2[N+]([O-])=O)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32N4O8S/c1-22-26(32-30(43-22)24-7-3-2-4-8-24)15-20-42-25-13-11-23(12-14-25)21-28(31(36)37)33-16-18-34(19-17-33)44(40,41)29-10-6-5-9-27(29)35(38)39/h2-14,28H,15-21H2,1H3,(H,36,37)/t28-/m0/s1
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n/an/an/an/a 2.16E+3n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM28681
PNG
(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Show SMILES CN(CCOc1ccc(Cc2sc(=O)[nH]c2O)cc1)c1ccccn1
Show InChI InChI=1S/C18H19N3O3S/c1-21(16-4-2-3-9-19-16)10-11-24-14-7-5-13(6-8-14)12-15-17(22)20-18(23)25-15/h2-9,22H,10-12H2,1H3,(H,20,23)
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n/an/an/an/a 35n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair		3D
3D Structure (crystal)
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50151001
PNG
((S)-2-((Z)-1-Methyl-3-oxo-3-phenyl-propenylamino)-...)
Show SMILES CC(CC(=O)c1ccccc1)=N[C@@H](Cc1ccc(OCCc2nc(oc2C)-c2ccccc2)cc1)C(O)=O |w:1.0|
Show InChI InChI=1S/C31H30N2O5/c1-21(19-29(34)24-9-5-3-6-10-24)32-28(31(35)36)20-23-13-15-26(16-14-23)37-18-17-27-22(2)38-30(33-27)25-11-7-4-8-12-25/h3-16,28H,17-20H2,1-2H3,(H,35,36)/t28-/m0/s1
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n/an/an/an/a 2.70n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315309
PNG
((S)-2-(4-(3-chlorophenyl)piperazin-1-yl)-3-(4-(2-(...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2cccc(Cl)c2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32ClN3O4/c1-22-28(33-30(39-22)24-6-3-2-4-7-24)14-19-38-27-12-10-23(11-13-27)20-29(31(36)37)35-17-15-34(16-18-35)26-9-5-8-25(32)21-26/h2-13,21,29H,14-20H2,1H3,(H,36,37)/t29-/m0/s1
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n/an/an/an/a>1.00E+5n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315308
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2ccc(C)cc2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C32H35N3O4/c1-23-8-12-27(13-9-23)34-17-19-35(20-18-34)30(32(36)37)22-25-10-14-28(15-11-25)38-21-16-29-24(2)39-31(33-29)26-6-4-3-5-7-26/h3-15,30H,16-22H2,1-2H3,(H,36,37)/t30-/m0/s1
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n/an/an/an/a 5.02E+4n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315312
PNG
((S)-2-(4-(2-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)S(=O)(=O)c2ccccc2F)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32FN3O6S/c1-22-27(33-30(41-22)24-7-3-2-4-8-24)15-20-40-25-13-11-23(12-14-25)21-28(31(36)37)34-16-18-35(19-17-34)42(38,39)29-10-6-5-9-26(29)32/h2-14,28H,15-21H2,1H3,(H,36,37)/t28-/m0/s1
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n/an/an/an/a 12n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315309
PNG
((S)-2-(4-(3-chlorophenyl)piperazin-1-yl)-3-(4-(2-(...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2cccc(Cl)c2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32ClN3O4/c1-22-28(33-30(39-22)24-6-3-2-4-7-24)14-19-38-27-12-10-23(11-13-27)20-29(31(36)37)35-17-15-34(16-18-35)26-9-5-8-25(32)21-26/h2-13,21,29H,14-20H2,1H3,(H,36,37)/t29-/m0/s1
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n/an/an/an/a 4.52E+4n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315308
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2ccc(C)cc2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C32H35N3O4/c1-23-8-12-27(13-9-23)34-17-19-35(20-18-34)30(32(36)37)22-25-10-14-28(15-11-25)38-21-16-29-24(2)39-31(33-29)26-6-4-3-5-7-26/h3-15,30H,16-22H2,1-2H3,(H,36,37)/t30-/m0/s1
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n/an/an/an/a>1.00E+5n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50151001
PNG
((S)-2-((Z)-1-Methyl-3-oxo-3-phenyl-propenylamino)-...)
Show SMILES CC(CC(=O)c1ccccc1)=N[C@@H](Cc1ccc(OCCc2nc(oc2C)-c2ccccc2)cc1)C(O)=O |w:1.0|
Show InChI InChI=1S/C31H30N2O5/c1-21(19-29(34)24-9-5-3-6-10-24)32-28(31(35)36)20-23-13-15-26(16-14-23)37-18-17-27-22(2)38-30(33-27)25-11-7-4-8-12-25/h3-16,28H,17-20H2,1-2H3,(H,35,36)/t28-/m0/s1
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n/an/an/an/a 10n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315310
PNG
((S)-3-(3-bromo-4-(2-(5-methyl-2-phenyloxazol-4-yl)...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2ccccc2)C(O)=O)cc1Br)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32BrN3O4/c1-22-27(33-30(39-22)24-8-4-2-5-9-24)14-19-38-29-13-12-23(20-26(29)32)21-28(31(36)37)35-17-15-34(16-18-35)25-10-6-3-7-11-25/h2-13,20,28H,14-19,21H2,1H3,(H,36,37)/t28-/m0/s1
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n/an/an/an/a>1.00E+5n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315313
PNG
((S)-2-(4-(4-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)S(=O)(=O)c2ccc(F)cc2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32FN3O6S/c1-22-28(33-30(41-22)24-5-3-2-4-6-24)15-20-40-26-11-7-23(8-12-26)21-29(31(36)37)34-16-18-35(19-17-34)42(38,39)27-13-9-25(32)10-14-27/h2-14,29H,15-21H2,1H3,(H,36,37)/t29-/m0/s1
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n/an/an/an/a 2.81E+3n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315306
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2cccc(C)c2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C32H35N3O4/c1-23-7-6-10-27(21-23)34-16-18-35(19-17-34)30(32(36)37)22-25-11-13-28(14-12-25)38-20-15-29-24(2)39-31(33-29)26-8-4-3-5-9-26/h3-14,21,30H,15-20,22H2,1-2H3,(H,36,37)/t30-/m0/s1
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n/an/an/an/a 8.98E+3n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM28681
PNG
(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Show SMILES CN(CCOc1ccc(Cc2sc(=O)[nH]c2O)cc1)c1ccccn1
Show InChI InChI=1S/C18H19N3O3S/c1-21(16-4-2-3-9-19-16)10-11-24-14-7-5-13(6-8-14)12-15-17(22)20-18(23)25-15/h2-9,22H,10-12H2,1H3,(H,20,23)
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n/an/an/an/a 1.06E+4n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315306
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2cccc(C)c2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C32H35N3O4/c1-23-7-6-10-27(21-23)34-16-18-35(19-17-34)30(32(36)37)22-25-11-13-28(14-12-25)38-20-15-29-24(2)39-31(33-29)26-8-4-3-5-9-26/h3-14,21,30H,15-20,22H2,1-2H3,(H,36,37)/t30-/m0/s1
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n/an/an/an/a 1.14E+3n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315307
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2ccccc2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H33N3O4/c1-23-28(32-30(38-23)25-8-4-2-5-9-25)16-21-37-27-14-12-24(13-15-27)22-29(31(35)36)34-19-17-33(18-20-34)26-10-6-3-7-11-26/h2-15,29H,16-22H2,1H3,(H,35,36)/t29-/m0/s1
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n/an/an/an/a 1.11E+4n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315310
PNG
((S)-3-(3-bromo-4-(2-(5-methyl-2-phenyloxazol-4-yl)...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2ccccc2)C(O)=O)cc1Br)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32BrN3O4/c1-22-27(33-30(39-22)24-8-4-2-5-9-24)14-19-38-29-13-12-23(20-26(29)32)21-28(31(36)37)35-17-15-34(16-18-35)25-10-6-3-7-11-25/h2-13,20,28H,14-19,21H2,1H3,(H,36,37)/t28-/m0/s1
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n/an/an/an/a>1.00E+5n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha


(Homo sapiens (Human))		BDBM50315311
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)S(=O)(=O)c2ccccc2[N+]([O-])=O)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H32N4O8S/c1-22-26(32-30(43-22)24-7-3-2-4-8-24)15-20-42-25-13-11-23(12-14-25)21-28(31(36)37)33-16-18-34(19-17-33)44(40,41)29-10-6-5-9-27(29)35(38)39/h2-14,28H,15-21H2,1H3,(H,36,37)/t28-/m0/s1
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n/an/an/an/a 1.45E+3n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma


(Homo sapiens (Human))		BDBM50315307
PNG
((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@H](N2CCN(CC2)c2ccccc2)C(O)=O)cc1)-c1ccccc1 |r|
Show InChI InChI=1S/C31H33N3O4/c1-23-28(32-30(38-23)25-8-4-2-5-9-25)16-21-37-27-14-12-24(13-15-27)22-29(31(35)36)34-19-17-33(18-20-34)26-10-6-3-7-11-26/h2-15,29H,16-22H2,1H3,(H,35,36)/t29-/m0/s1
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n/an/an/an/a 1.06E+4n/an/an/an/a



Institute of Pharmacology and Toxicology

Curated by ChEMBL


Assay Description
Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assay

Bioorg Med Chem Lett 20: 2605-8 (2010)


Article DOI: 10.1016/j.bmcl.2010.02.071
BindingDB Entry DOI: 10.7270/Q2HD7WMW
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%