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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Transcription factor Jun (Homo sapiens (Human)) | BDBM50315777 (3-(4-Acetyl-phenyl)-2-(5-morpholin-4-yl-4-pyridin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
B. V. Patel Pharmaceutical Education and Research Development Centre Curated by ChEMBL | Assay Description Inhibition of AP-1 expressed in HEK293 cells assessed as PMA-stimulated transcriptional activation treated 24 hrs before PMA challenge measured after... | Bioorg Med Chem 18: 2796-808 (2010) Article DOI: 10.1016/j.bmc.2010.01.007 BindingDB Entry DOI: 10.7270/Q2S182NG | |||||||||||
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