Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50316544 (3-((6-chlorothiazolo[4,5-b]pyridin-2-yl)methoxy)-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Biota Europe Ltd. Curated by ChEMBL | Assay Description Inhibition of human ERG by single cell patch-clamp assay | J Med Chem 53: 3927-36 (2010) Article DOI: 10.1021/jm9016366 BindingDB Entry DOI: 10.7270/Q2K64J77 | |||||||||||
More data for this Ligand-Target Pair |