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PubMed code 20483601

Compile data set for download or QSAR
Found 22 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320090
PNG
((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Show SMILES CN(CC1CC1)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@H](c23)[C@@]1(O)CCC4=O |r|
Show InChI InChI=1S/C19H23NO4/c1-20(9-10-2-3-10)14-8-11-4-5-12(21)17-15(11)16-18(24-17)13(22)6-7-19(14,16)23/h4-5,10,14,16,18,21,23H,2-3,6-9H2,1H3/t14-,16+,18+,19-/m1/s1
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 1.17n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320086
PNG
((2R,2aR,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Show SMILES CN(CC1CC1)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@@H]([C@H]1CCC4=O)c23 |r|
Show InChI InChI=1S/C19H23NO3/c1-20(9-10-2-3-10)13-8-11-4-6-14(21)18-16(11)17-12(13)5-7-15(22)19(17)23-18/h4,6,10,12-13,17,19,21H,2-3,5,7-9H2,1H3/t12-,13+,17-,19-/m0/s1
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 3.36n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320090
PNG
((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Show SMILES CN(CC1CC1)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@H](c23)[C@@]1(O)CCC4=O |r|
Show InChI InChI=1S/C19H23NO4/c1-20(9-10-2-3-10)14-8-11-4-5-12(21)17-15(11)16-18(24-17)13(22)6-7-19(14,16)23/h4-5,10,14,16,18,21,23H,2-3,6-9H2,1H3/t14-,16+,18+,19-/m1/s1
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 5.10n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320086
PNG
((2R,2aR,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Show SMILES CN(CC1CC1)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@@H]([C@H]1CCC4=O)c23 |r|
Show InChI InChI=1S/C19H23NO3/c1-20(9-10-2-3-10)13-8-11-4-6-14(21)18-16(11)17-12(13)5-7-15(22)19(17)23-18/h4,6,10,12-13,17,19,21H,2-3,5,7-9H2,1H3/t12-,13+,17-,19-/m0/s1
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 8.81n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320089
PNG
((2R,2aS,2a1S,5aR)-2-(dimethylamino)-2a,7-dihydroxy...)
Show SMILES CN(C)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@H](c23)[C@@]1(O)CCC4=O |r|
Show InChI InChI=1S/C16H19NO4/c1-17(2)11-7-8-3-4-9(18)14-12(8)13-15(21-14)10(19)5-6-16(11,13)20/h3-4,11,13,15,18,20H,5-7H2,1-2H3/t11-,13+,15+,16-/m1/s1
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 8.95n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320088
PNG
((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a,7-...)
Show SMILES Oc1ccc2C[C@@H](NCC3CC3)[C@]3(O)CCC(=O)[C@@H]4Oc1c2[C@H]34 |r|
Show InChI InChI=1S/C18H21NO4/c20-11-4-3-10-7-13(19-8-9-1-2-9)18(22)6-5-12(21)17-15(18)14(10)16(11)23-17/h3-4,9,13,15,17,19-20,22H,1-2,5-8H2/t13-,15+,17+,18-/m1/s1
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 24.7n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320084
PNG
((2R,2aR,2a1S,5aR)-2-(cyclopropylmethylamino)-7-hyd...)
Show SMILES Oc1ccc2C[C@@H](NCC3CC3)[C@@H]3CCC(=O)[C@@H]4Oc1c2[C@H]34 |r|
Show InChI InChI=1S/C18H21NO3/c20-13-5-3-10-7-12(19-8-9-1-2-9)11-4-6-14(21)18-16(11)15(10)17(13)22-18/h3,5,9,11-12,16,18-20H,1-2,4,6-8H2/t11-,12+,16-,18-/m0/s1
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 30.3n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320084
PNG
((2R,2aR,2a1S,5aR)-2-(cyclopropylmethylamino)-7-hyd...)
Show SMILES Oc1ccc2C[C@@H](NCC3CC3)[C@@H]3CCC(=O)[C@@H]4Oc1c2[C@H]34 |r|
Show InChI InChI=1S/C18H21NO3/c20-13-5-3-10-7-12(19-8-9-1-2-9)11-4-6-14(21)18-16(11)15(10)17(13)22-18/h3,5,9,11-12,16,18-20H,1-2,4,6-8H2/t11-,12+,16-,18-/m0/s1
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 32.2n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320085
PNG
((2R,2aR,2a1S,5aR)-2-(dimethylamino)-7-hydroxy-2,2a...)
Show SMILES CN(C)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@@H]([C@H]1CCC4=O)c23 |r|
Show InChI InChI=1S/C16H19NO3/c1-17(2)10-7-8-3-5-11(18)15-13(8)14-9(10)4-6-12(19)16(14)20-15/h3,5,9-10,14,16,18H,4,6-7H2,1-2H3/t9-,10+,14-,16-/m0/s1
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 50.9n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320088
PNG
((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a,7-...)
Show SMILES Oc1ccc2C[C@@H](NCC3CC3)[C@]3(O)CCC(=O)[C@@H]4Oc1c2[C@H]34 |r|
Show InChI InChI=1S/C18H21NO4/c20-11-4-3-10-7-13(19-8-9-1-2-9)18(22)6-5-12(21)17-15(18)14(10)16(11)23-17/h3-4,9,13,15,17,19-20,22H,1-2,5-8H2/t13-,15+,17+,18-/m1/s1
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 68.4n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320093
PNG
((1S,5R,13S,20R)-8-hydroxy-6,19-dioxa-16-azahexacyc...)
Show SMILES Oc1ccc2C[C@H]3N4CCO[C@]33CCC(=O)[C@@H]5Oc1c2[C@]35CC4 |r,TLB:19:20:6:10.8.9,THB:16:20:6:10.8.9|
Show InChI InChI=1S/C18H19NO4/c20-11-2-1-10-9-13-18-4-3-12(21)16-17(18,14(10)15(11)23-16)5-6-19(13)7-8-22-18/h1-2,13,16,20H,3-9H2/t13-,16+,17+,18-/m1/s1
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 72.6n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320093
PNG
((1S,5R,13S,20R)-8-hydroxy-6,19-dioxa-16-azahexacyc...)
Show SMILES Oc1ccc2C[C@H]3N4CCO[C@]33CCC(=O)[C@@H]5Oc1c2[C@]35CC4 |r,TLB:19:20:6:10.8.9,THB:16:20:6:10.8.9|
Show InChI InChI=1S/C18H19NO4/c20-11-2-1-10-9-13-18-4-3-12(21)16-17(18,14(10)15(11)23-16)5-6-19(13)7-8-22-18/h1-2,13,16,20H,3-9H2/t13-,16+,17+,18-/m1/s1
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 86n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320087
PNG
((2R,2aS,2a1S,5aR)-2a,7-dihydroxy-2-(methylamino)-2...)
Show SMILES CN[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@H](c23)[C@@]1(O)CCC4=O |r|
Show InChI InChI=1S/C15H17NO4/c1-16-10-6-7-2-3-8(17)13-11(7)12-14(20-13)9(18)4-5-15(10,12)19/h2-3,10,12,14,16-17,19H,4-6H2,1H3/t10-,12+,14+,15-/m1/s1
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 118n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320083
PNG
((2R,2aR,2a1S,5aR)-7-hydroxy-2-(methylamino)-2,2a,2...)
Show SMILES CN[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@@H]([C@H]1CCC4=O)c23 |r|
Show InChI InChI=1S/C15H17NO3/c1-16-9-6-7-2-4-10(17)14-12(7)13-8(9)3-5-11(18)15(13)19-14/h2,4,8-9,13,15-17H,3,5-6H2,1H3/t8-,9+,13-,15-/m0/s1
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 164n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320091
PNG
((1R,5S,10R,18S)-9-(cyclopropylmethyl)-15-hydroxy-6...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CCO[C@]33CCC(=O)[C@@H]4Oc1c2[C@H]34 |r|
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24-8-7-21(15)10-11-1-2-11)6-5-14(23)19-17(20)16(12)18(13)25-19/h3-4,11,15,17,19,22H,1-2,5-10H2/t15-,17+,19+,20-/m1/s1
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 294n/an/an/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320092
PNG
((1R,5S,10R,18S)-15-hydroxy-9-methyl-6,19-dioxa-9-a...)
Show SMILES CN1CCO[C@@]23CCC(=O)[C@@H]4Oc5c([C@H]24)c(C[C@@H]13)ccc5O |r|
Show InChI InChI=1S/C17H19NO4/c1-18-6-7-21-17-5-4-11(20)16-14(17)13-9(8-12(17)18)2-3-10(19)15(13)22-16/h2-3,12,14,16,19H,4-8H2,1H3/t12-,14+,16+,17-/m1/s1
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n/an/a>1.00E+3n/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320089
PNG
((2R,2aS,2a1S,5aR)-2-(dimethylamino)-2a,7-dihydroxy...)
Show SMILES CN(C)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@H](c23)[C@@]1(O)CCC4=O |r|
Show InChI InChI=1S/C16H19NO4/c1-17(2)11-7-8-3-4-9(18)14-12(8)13-15(21-14)10(19)5-6-16(11,13)20/h3-4,11,13,15,18,20H,5-7H2,1-2H3/t11-,13+,15+,16-/m1/s1
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n/an/a>1.00E+3n/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320087
PNG
((2R,2aS,2a1S,5aR)-2a,7-dihydroxy-2-(methylamino)-2...)
Show SMILES CN[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@H](c23)[C@@]1(O)CCC4=O |r|
Show InChI InChI=1S/C15H17NO4/c1-16-10-6-7-2-3-8(17)13-11(7)12-14(20-13)9(18)4-5-15(10,12)19/h2-3,10,12,14,16-17,19H,4-6H2,1H3/t10-,12+,14+,15-/m1/s1
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n/an/a>1.00E+3n/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320091
PNG
((1R,5S,10R,18S)-9-(cyclopropylmethyl)-15-hydroxy-6...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CCO[C@]33CCC(=O)[C@@H]4Oc1c2[C@H]34 |r|
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24-8-7-21(15)10-11-1-2-11)6-5-14(23)19-17(20)16(12)18(13)25-19/h3-4,11,15,17,19,22H,1-2,5-10H2/t15-,17+,19+,20-/m1/s1
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n/an/a>1.00E+3n/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50320092
PNG
((1R,5S,10R,18S)-15-hydroxy-9-methyl-6,19-dioxa-9-a...)
Show SMILES CN1CCO[C@@]23CCC(=O)[C@@H]4Oc5c([C@H]24)c(C[C@@H]13)ccc5O |r|
Show InChI InChI=1S/C17H19NO4/c1-18-6-7-21-17-5-4-11(20)16-14(17)13-9(8-12(17)18)2-3-10(19)15(13)22-16/h2-3,12,14,16,19H,4-8H2,1H3/t12-,14+,16+,17-/m1/s1
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n/an/a>1.00E+3n/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation counting

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320085
PNG
((2R,2aR,2a1S,5aR)-2-(dimethylamino)-7-hydroxy-2,2a...)
Show SMILES CN(C)[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@@H]([C@H]1CCC4=O)c23 |r|
Show InChI InChI=1S/C16H19NO3/c1-17(2)10-7-8-3-5-11(18)15-13(8)14-9(10)4-6-12(19)16(14)20-15/h3,5,9-10,14,16,18H,4,6-7H2,1-2H3/t9-,10+,14-,16-/m0/s1
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Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50320083
PNG
((2R,2aR,2a1S,5aR)-7-hydroxy-2-(methylamino)-2,2a,2...)
Show SMILES CN[C@@H]1Cc2ccc(O)c3O[C@@H]4[C@@H]([C@H]1CCC4=O)c23 |r|
Show InChI InChI=1S/C15H17NO3/c1-16-9-6-7-2-4-10(17)14-12(7)13-8(9)3-5-11(18)15(13)19-14/h2,4,8-9,13,15-17H,3,5-6H2,1H3/t8-,9+,13-,15-/m0/s1
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n/an/a>1.00E+3n/an/an/an/an/an/a



Kitasato University

Curated by ChEMBL


Assay Description
Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counter

Bioorg Med Chem Lett 20: 3726-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.04.080
BindingDB Entry DOI: 10.7270/Q2KD1Z3B
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%