Affinity Data by PubMed id=20667726

PubMed code 20667726

Found 3 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50325039 (6-(ethyl(1-isobutyl-2-oxo-4-(trifluoromethyl)-1,2-...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a
Okayama University Curated by ChEMBL					Assay Description Agonist activity at human RXRalpha expressed in human COS7 cells by luciferase reporter gene assay				Bioorg Med Chem Lett 20: 5143-6 (2010) Article DOI: 10.1016/j.bmcl.2010.07.011 BindingDB Entry DOI: 10.7270/Q2ZG6SG6
Okayama University Curated by ChEMBL					More data for this Ligand-Target Pair
Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50325038 (6-(ethyl(8-ethyl-7-oxo-5-(trifluoromethyl)-7,8-dih...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a
Okayama University Curated by ChEMBL					Assay Description Agonist activity at human RXRalpha expressed in human COS7 cells by luciferase reporter gene assay				Bioorg Med Chem Lett 20: 5143-6 (2010) Article DOI: 10.1016/j.bmcl.2010.07.011 BindingDB Entry DOI: 10.7270/Q2ZG6SG6
Okayama University Curated by ChEMBL					More data for this Ligand-Target Pair
Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50325037 (6-(ethyl(8-methyl-7-oxo-5-(trifluoromethyl)-7,8-di...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a
Okayama University Curated by ChEMBL					Assay Description Agonist activity at human RXRalpha expressed in human COS7 cells by luciferase reporter gene assay				Bioorg Med Chem Lett 20: 5143-6 (2010) Article DOI: 10.1016/j.bmcl.2010.07.011 BindingDB Entry DOI: 10.7270/Q2ZG6SG6
Okayama University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%