Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Retinoic acid receptor RXR-alpha (Homo sapiens (Human)) | BDBM50157304 (3',5-di-2-propenyl-1,1'-biphenyl-2,4'-diol | 3',5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.18E+4 | n/a | n/a | n/a | n/a |
Aichi Gakuin University Curated by ChEMBL | Assay Description Agonist activity at RXRalpha in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter gene assay | J Nat Prod 73: 1332-6 (2010) Article DOI: 10.1021/np100120c BindingDB Entry DOI: 10.7270/Q2VT1S9K | |||||||||||
More data for this Ligand-Target Pair |