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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50343035 (4,5,6,7-Tetrachloro-N-{3-[2-(3-trifluoromethylphen...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Inhibition of DPP4 assessed as p-nitrophenol release after 1 hr | Bioorg Med Chem Lett 21: 3041-5 (2011) Article DOI: 10.1016/j.bmcl.2011.03.026 BindingDB Entry DOI: 10.7270/Q2RR1ZKM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50343036 (4,5,6,7-Tetrachloro-N-{3-[2-(2-trifluoromethylphen...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Inhibition of DPP4 assessed as p-nitrophenol release after 1 hr | Bioorg Med Chem Lett 21: 3041-5 (2011) Article DOI: 10.1016/j.bmcl.2011.03.026 BindingDB Entry DOI: 10.7270/Q2RR1ZKM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Dipeptidyl peptidase 8 (Homo sapiens (Human)) | BDBM50343036 (4,5,6,7-Tetrachloro-N-{3-[2-(2-trifluoromethylphen...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Inhibition of DPP8 assessed as p-nitrophenol release after 1 hr | Bioorg Med Chem Lett 21: 3041-5 (2011) Article DOI: 10.1016/j.bmcl.2011.03.026 BindingDB Entry DOI: 10.7270/Q2RR1ZKM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Dipeptidyl peptidase 8 (Homo sapiens (Human)) | BDBM50343034 (4,5,6,7-Tetrachloro-N-{3-[2-(4-trifluoromethylphen...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Inhibition of DPP8 assessed as p-nitrophenol release after 1 hr | Bioorg Med Chem Lett 21: 3041-5 (2011) Article DOI: 10.1016/j.bmcl.2011.03.026 BindingDB Entry DOI: 10.7270/Q2RR1ZKM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Dipeptidyl peptidase 8 (Homo sapiens (Human)) | BDBM50298687 (4,5,6,7-Tetrachloro-N-[3-(2-phenylethyl)phenyl]pht...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Inhibition of DPP8 assessed as p-nitrophenol release after 1 hr | Bioorg Med Chem Lett 21: 3041-5 (2011) Article DOI: 10.1016/j.bmcl.2011.03.026 BindingDB Entry DOI: 10.7270/Q2RR1ZKM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Dipeptidyl peptidase 8 (Homo sapiens (Human)) | BDBM50343035 (4,5,6,7-Tetrachloro-N-{3-[2-(3-trifluoromethylphen...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Inhibition of DPP8 assessed as p-nitrophenol release after 1 hr | Bioorg Med Chem Lett 21: 3041-5 (2011) Article DOI: 10.1016/j.bmcl.2011.03.026 BindingDB Entry DOI: 10.7270/Q2RR1ZKM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
