Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50265534 (2-((2R,8R,11R,14S)-11-(4-aminobutyl)-8-(3-guanidin...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 116 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Delaware Curated by ChEMBL | Assay Description Displacement of [125]I-echistatin from alphaVbeta3 integrin expressed in human U87MG cells by competitive binding assay | Bioorg Med Chem Lett 21: 5011-4 (2011) Article DOI: 10.1016/j.bmcl.2011.04.116 BindingDB Entry DOI: 10.7270/Q2319X5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-V/beta-3 (Homo sapiens (Human)) | BDBM50419042 (CHEMBL1824706) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 193 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Delaware Curated by ChEMBL | Assay Description Displacement of [125]I-echistatin from alphaVbeta3 integrin expressed in human U87MG cells by competitive binding assay | Bioorg Med Chem Lett 21: 5011-4 (2011) Article DOI: 10.1016/j.bmcl.2011.04.116 BindingDB Entry DOI: 10.7270/Q2319X5Q | |||||||||||
More data for this Ligand-Target Pair |